Azoles

cytochrome P450 family 19 subfamily A member 1 ; Homo sapiens







9 Article(s)
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Title
Pub. Year
#Total Relationships
1 35176449 Exploration of structural requirements for azole chemicals towards human aromatase CYP19A1 activity: Classification modeling, structure-activity relationships and read-across study. 2022 Jun 2
2 32046297 Towards an Understanding of the Mode of Action of Human Aromatase Activity for Azoles through Quantum Chemical Descriptors-Based Regression and Structure Activity Relationship Modeling Analysis. 2020 Feb 8 3
3 32435378 Targeting Orthosteric and Allosteric Pockets of Aromatase via Dual-Mode Novel Azole Inhibitors. 2020 May 14 2
4 31330226 The classic azole antifungal drugs are highly potent endocrine disruptors in vitro inhibiting steroidogenic CYP enzymes at concentrations lower than therapeutic Cmax. 2019 Sep 1 1
5 24274332 Human and ecological risk assessment of a crop protection chemical: a case study with the azole fungicide epoxiconazole. 2014 Feb 1
6 19500885 An efficient steroid pharmacophore-based strategy to identify new aromatase inhibitors. 2009 Oct 1
7 16330141 Inhibition of human CYP19 by azoles used as antifungal agents and aromatase inhibitors, using a new LC-MS/MS method for the analysis of estradiol product formation. 2006 Feb 15 3
8 15380230 Synthesis and evaluation of 4-triazolylflavans as new aromatase inhibitors. 2004 Oct 18 1
9 15554355 Comparative assessment of the inhibition of recombinant human CYP19 (aromatase) by azoles used in agriculture and as drugs for humans. 2004 Aug 3