| 1 |
29872302 | Valium without dependence? Individual GABAA receptor subtype contribution toward benzodiazepine addiction, tolerance, and therapeutic effects. | 2018 |
1 |
| 2 |
30210295 | Distinct Modulation of Spontaneous and GABA-Evoked Gating by Flurazepam Shapes Cross-Talk Between Agonist-Free and Liganded GABAA Receptor Activity. | 2018 |
1 |
| 3 |
28445782 | The immunohistochemical distribution of the GABAA receptor α1, α2, α3, β2/3 and γ2 subunits in the human thalamus. | 2017 Jul |
1 |
| 4 |
29138471 | α subunits in GABAA receptors are dispensable for GABA and diazepam action. | 2017 Nov 14 |
2 |
| 5 |
23088350 | A prospective test of the late effects of potentially antineuroplastic drugs in a stroke rehabilitation study. | 2014 Jun |
1 |
| 6 |
24241181 | Some insights into the binding mechanism of the GABAA receptor: a combined docking and MM-GBSA study. | 2013 Dec |
4 |
| 7 |
20417252 | Human locus coeruleus neurons express the GABA(A) receptor gamma2 subunit gene and produce benzodiazepine binding. | 2010 Jun 21 |
1 |
| 8 |
21309116 | GABAA receptor alpha2/alpha3 subtype-selective modulators as potential nonsedating anxiolytics. | 2010 |
1 |
| 9 |
17539703 | Mechanisms of sleep induction by GABA(A) receptor agonists. | 2007 |
1 |
| 10 |
17953656 | Replacement of histidine in position 105 in the α₅ subunit by cysteine stimulates zolpidem sensitivity of α₅β₂γ₂ GABA(A) receptors. | 2007 Dec |
2 |
| 11 |
19300612 | Indiplon in the treatment of sleep disorders. | 2007 Dec |
1 |
| 12 |
15926867 | The benzodiazepine binding site of GABA(A) receptors as a target for the development of novel anxiolytics. | 2005 May |
2 |
| 13 |
15125950 | 3,4-Dihydronaphthalen-1(2H)-ones: novel ligands for the benzodiazepine site of alpha5-containing GABAA receptors. | 2004 Jun 7 |
1 |
| 14 |
15505688 | [New molecular targets in pharmacological treatment of anxiety disorders]. | 2004 |
2 |
| 15 |
12871032 | Anxioselective compounds acting at the GABA(A) receptor benzodiazepine binding site. | 2003 Aug |
1 |
| 16 |
14573876 | Recombinant extracellular domain of the three major subunits of GABAA receptor show comparable secondary structure and benzodiazepine binding properties. | 2003 Nov |
4 |
| 17 |
12171574 | Mapping of the benzodiazepine recognition site on GABA(A) receptors. | 2002 Aug |
1 |
| 18 |
11299307 | Identification of amino acid residues responsible for the alpha5 subunit binding selectivity of L-655,708, a benzodiazepine binding site ligand at the GABA(A) receptor. | 2001 Apr |
1 |
| 19 |
11306694 | Effect of alpha subunit on allosteric modulation of ion channel function in stably expressed human recombinant gamma-aminobutyric acid(A) receptors determined using (36)Cl ion flux. | 2001 May |
1 |
| 20 |
11595770 | Prevalence between different alpha subunits performing the benzodiazepine binding sites in native heterologous GABA(A) receptors containing the alpha2 subunit. | 2001 Oct |
1 |
| 21 |
11100148 | Benzodiazepines act on GABAA receptors via two distinct and separable mechanisms. | 2000 Dec |
2 |
| 22 |
10224099 | Structural elements of the gamma-aminobutyric acid type A receptor conferring subtype selectivity for benzodiazepine site ligands. | 1999 May 7 |
1 |
| 23 |
10501225 | Role of the conserved lysine residue in the middle of the predicted extracellular loop between M2 and M3 in the GABA(A) receptor. | 1999 Oct |
1 |
| 24 |
9652349 | Regulation of GABA(A) receptor alpha1 protein is a sensitive indicator of benzodiazepine agonist efficacy. | 1998 May 8 |
2 |
| 25 |
9754930 | Amino acid residue 200 on the alpha1 subunit of GABA(A) receptors affects the interaction with selected benzodiazepine binding site ligands. | 1998 Aug 7 |
1 |
| 26 |
8592140 | The alpha 1 and alpha 6 subunits can coexist in the same cerebellar GABAA receptor maintaining their individual benzodiazepine-binding specificities. | 1996 Feb |
4 |
| 27 |
8723715 | Striatal efferents preferentially innervate neurons in the ventral pallidum containing GABAA receptor alpha 1 subunit-like immunoreactivity. | 1996 Jun |
2 |
| 28 |
7780638 | Interaction of beta-carboline inverse agonists for the benzodiazepine site with another site on GABAA receptors. | 1995 Mar |
1 |
| 29 |
7799410 | Four amino acid exchanges convert a diazepam-insensitive, inverse agonist-preferring GABAA receptor into a diazepam-preferring GABAA receptor. | 1994 Dec 23 |
1 |
| 30 |
7901754 | Potentiation of gamma-aminobutyric acid-induced chloride currents by various benzodiazepine site agonists with the alpha 1 gamma 2, beta 2 gamma 2 and alpha 1 beta 2 gamma 2 subtypes of cloned gamma-aminobutyric acid type A receptors. | 1993 Oct |
7 |
| 31 |
8242240 | Differential affinity of dihydroimidazoquinoxalines and diimidazoquinazolines to the alpha 1 beta 2 gamma 2 and alpha 6 beta 2 gamma 2 subtypes of cloned GABAA receptors. | 1993 Oct |
2 |
| 32 |
8391122 | Cloning of cDNA sequences encoding human alpha 2 and alpha 3 gamma-aminobutyric acidA receptor subunits and characterization of the benzodiazepine pharmacology of recombinant alpha 1-, alpha 2-, alpha 3-, and alpha 5-containing human gamma-aminobutyric acidA receptors. | 1993 Jun |
1 |
| 33 |
1321437 | Stable expression of mammalian type A gamma-aminobutyric acid receptors in mouse cells: demonstration of functional assembly of benzodiazepine-responsive sites. | 1992 Jul 15 |
1 |
| 34 |
1346133 | A single histidine in GABAA receptors is essential for benzodiazepine agonist binding. | 1992 Jan 25 |
3 |
| 35 |
1664058 | The GABAA receptor family in the mammalian brain. | 1991 Mar |
1 |
| 36 |
1665550 | Inverse but not full benzodiazepine agonists modulate recombinant alpha 6 beta 2 gamma 2 GABAA receptors in transfected human embryonic kidney cells. | 1991 Sep 16 |
1 |