| 1 |
34847409 | Application of the dual-tail approach for the design and synthesis of novel Thiopyrimidine-Benzenesulfonamide hybrids as selective carbonic anhydrase inhibitors. | 2022 Jan 15 |
2 |
| 2 |
33472371 | Modulation of the Pharmacokinetics of a Radioligand Targeting Carbonic Anhydrase-IX with Albumin-Binding Moieties. | 2021 Mar 1 |
1 |
| 3 |
33523653 | Inhibition of Carbonic Anhydrase Using SLC-149: Support for a Noncatalytic Function of CAIX in Breast Cancer. | 2021 Feb 11 |
1 |
| 4 |
33905156 | Affinity Selections of DNA-Encoded Chemical Libraries on Carbonic Anhydrase IX-Expressing Tumor Cells Reveal a Dependence on Ligand Valence. | 2021 Jun 21 |
1 |
| 5 |
34138317 | Targeting Hypoxic Tumors with Hybrid Nanobullets for Oxygen-Independent Synergistic Photothermal and Thermodynamic Therapy. | 2021 Mar 31 |
4 |
| 6 |
34443307 | Design, Synthesis, Biological Evaluation, and Computational Studies of Novel Tri-Aryl Imidazole-Benzene Sulfonamide Hybrids as Promising Selective Carbonic Anhydrase IX and XII Inhibitors. | 2021 Aug 4 |
1 |
| 7 |
34450241 | A novel 111indium-labeled dual carbonic anhydrase 9-targeted probe as a potential SPECT imaging radiotracer for detection of hypoxic colorectal cancer cells. | 2021 Nov |
5 |
| 8 |
33085484 | Structural Basis of Nanomolar Inhibition of Tumor-Associated Carbonic Anhydrase IX: X-Ray Crystallographic and Inhibition Study of Lipophilic Inhibitors with Acetazolamide Backbone. | 2020 Nov 12 |
2 |
| 9 |
30746618 | Carbonic anhydrase-IX inhibition enhances the efficacy of hexokinase II inhibitor for hepatocellular carcinoma in a murine model. | 2019 Apr |
1 |
| 10 |
30892905 | Development of the 99mTc-Hydroxamamide Complex as a Probe Targeting Carbonic Anhydrase IX. | 2019 Apr 1 |
1 |
| 11 |
31590289 | Extending the Inhibition Profiles of Coumarin-Based Compounds Against Human Carbonic Anhydrases: Synthesis, Biological, and In Silico Evaluation. | 2019 Oct 4 |
1 |
| 12 |
31667562 | Automated and enhanced extraction of a small molecule-drug conjugate using an enzyme-inhibitor interaction based SPME tool followed by direct analysis by ESI-MS. | 2019 Nov |
2 |
| 13 |
29422388 | Acetazolamide-based [18F]-PET tracer: In vivo validation of carbonic anhydrase IX as a sole target for imaging of CA-IX expressing hypoxic solid tumors. | 2018 Mar 1 |
6 |
| 14 |
29534020 | Copper-Free 'Click' Chemistry-Based Synthesis and Characterization of Carbonic Anhydrase-IX Anchored Albumin-Paclitaxel Nanoparticles for Targeting Tumor Hypoxia. | 2018 Mar 13 |
2 |
| 15 |
29929883 | Corrigendum to "Acetazolamide-based [18F]-PET tracer: In vivo validation of carbonic anhydrase IX as a sole target for imaging of CA-IX expressing hypoxic solid tumors" [Bioorg. Med. Chem. Lett. 28 (5) (2018) 915-921]. | 2018 Aug 1 |
2 |
| 16 |
30153589 | Novel sulfonamides incorporating 1,3,5-triazine and amino acid structural motifs as inhibitors of the physiological carbonic anhydrase isozymes I, II and IV and tumor-associated isozyme IX. | 2018 Dec |
1 |
| 17 |
30185025 | Carbonic Anhydrase IX-Targeted Near-Infrared Dye for Fluorescence Imaging of Hypoxic Tumors. | 2018 Oct 17 |
2 |
| 18 |
30533574 | In Vivo Antitumor Activity of a Novel Acetazolamide-Cryptophycin Conjugate for the Treatment of Renal Cell Carcinomas. | 2018 Nov 30 |
1 |
| 19 |
27373313 | Virtual screening, molecular dynamics, and binding free energy calculations on human carbonic anhydrase IX catalytic domain for deciphering potential leads. | 2017 Aug |
2 |
| 20 |
27890855 | Linker stability influences the anti-tumor activity of acetazolamide-drug conjugates for the therapy of renal cell carcinoma. | 2017 Jan 28 |
2 |
| 21 |
28067010 | Hit-Validation Methodologies for Ligands Isolated from DNA-Encoded Chemical Libraries. | 2017 May 4 |
1 |
| 22 |
28520445 | Telodendrimers for Physical Encapsulation and Covalent Linking of Individual or Combined Therapeutics. | 2017 Aug 7 |
1 |
| 23 |
28943245 | Improved molecular recognition of Carbonic Anhydrase IX by polypeptide conjugation to acetazolamide. | 2017 Oct 15 |
2 |
| 24 |
27609641 | Acetazolamide Serves as Selective Delivery Vehicle for Dipeptide-Linked Drugs to Renal Cell Carcinoma. | 2016 Dec |
3 |
| 25 |
27702686 | Inhibition of carbonic anhydrase IX in glioblastoma multiforme. | 2016 Dec |
2 |
| 26 |
25711495 | Synthesis of sulfonamide conjugates of Cu(II), Ga(III), In(III), Re(V) and Zn(II) complexes: carbonic anhydrase inhibition studies and cellular imaging investigations. | 2015 Mar 21 |
1 |
| 27 |
25793203 | Binding of carbonic anhydrase IX to 45S rDNA genes is prevented by exportin-1 in hypoxic cells. | 2015 |
1 |
| 28 |
26522624 | Efficient Expression and Crystallization System of Cancer-Associated Carbonic Anhydrase Isoform IX. | 2015 Nov 25 |
1 |
| 29 |
23163664 | Inhibition of carbonic anhydrase activity modifies the toxicity of doxorubicin and melphalan in tumour cells in vitro. | 2013 Apr |
2 |
| 30 |
23706268 | Hypoxia induced CA9 inhibitory targeting by two different sulfonamide derivatives including acetazolamide in human glioblastoma. | 2013 Jul 1 |
2 |
| 31 |
21676479 | Specific inhibition of carbonic anhydrase IX activity enhances the in vivo therapeutic effect of tumor irradiation. | 2011 Jun |
1 |
| 32 |
19170619 | Design of a carbonic anhydrase IX active-site mimic to screen inhibitors for possible anticancer properties. | 2009 Feb 17 |
1 |
| 33 |
19615903 | In vivo targeting of tumor-associated carbonic anhydrases using acetazolamide derivatives. | 2009 Aug 15 |
1 |
| 34 |
19805286 | Crystal structure of the catalytic domain of the tumor-associated human carbonic anhydrase IX. | 2009 Sep 22 |
1 |
| 35 |
18295485 | Carbonic anhydrase inhibitors: the very weak inhibitors dithiothreitol, beta-mercaptoethanol, tris(carboxyethyl)phosphine and threitol interfere with the binding of sulfonamides to isozymes II and IX. | 2008 Mar 15 |
2 |
| 36 |
16165351 | Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with benzo[b]thiophene 1,1-dioxide sulfonamides. | 2005 Nov 1 |
1 |
| 37 |
12643899 | Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with aromatic and heterocyclic sulfonamides. | 2003 Mar 24 |
1 |