| 1 |
35616541 | Anticancer carbonic anhydrase inhibitors: a patent and literature update 2018-2022. | 2022 Jun 2 |
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| 2 |
34198834 | Inhibition of Carbonic Anhydrase IX Promotes Apoptosis through Intracellular pH Level Alterations in Cervical Cancer Cells. | 2021 Jun 5 |
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| 3 |
34445506 | Betulin Sulfonamides as Carbonic Anhydrase Inhibitors and Anticancer Agents in Breast Cancer Cells. | 2021 Aug 16 |
2 |
| 4 |
34948406 | Synthesis, Molecular Docking Analysis, and Biological Evaluations of Saccharide-Modified Sulfonamides as Carbonic Anhydrase IX Inhibitors. | 2021 Dec 19 |
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| 5 |
31718943 | Synthesis, biological and molecular dynamics investigations with a series of triazolopyrimidine/triazole-based benzenesulfonamides as novel carbonic anhydrase inhibitors. | 2020 Jan 1 |
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| 6 |
31915112 | Benzimidazole derivatives as potent and isoform selective tumor-associated carbonic anhydrase IX/XII inhibitors. | 2020 Jan |
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| 7 |
32044580 | Inclusion of a 5-fluorouracil moiety in nitrogenous bases derivatives as human carbonic anhydrase IX and XII inhibitors produced a targeted action against MDA-MB-231 and T47D breast cancer cells. | 2020 Mar 15 |
2 |
| 8 |
32182519 | Appliance of the piperidinyl-hydrazidoureido linker to benzenesulfonamide compounds: Synthesis, in vitro and in silico evaluation of potent carbonic anhydrase II, IX and XII inhibitors. | 2020 May |
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| 9 |
32340282 | Pharmacological Inhibition of CA-IX Impairs Tumor Cell Proliferation, Migration and Invasiveness. | 2020 Apr 23 |
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| 10 |
32891000 | Pyridinium derivatives of 3-aminobenzenesulfonamide are nanomolar-potent inhibitors of tumor-expressed carbonic anhydrase isozymes CA IX and CA XII. | 2020 Oct |
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| 11 |
32911194 | Design, synthesis and biological evaluation of novel carbohydrate-based sulfonamide derivatives as antitumor agents. | 2020 Nov |
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| 12 |
33142414 | Discovery of novel artemisinin-sulfonamidehybrids as potential carbonicanhydraseIX inhibitors with improved antiproliferative activities. | 2020 Nov |
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| 13 |
33159147 | In vitro and in vivo BNCT investigations using a carborane containing sulfonamide targeting CAIX epitopes on malignant pleural mesothelioma and breast cancer cells. | 2020 Nov 6 |
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| 14 |
30978604 | Novel synthesized SLC-0111 thiazole and thiadiazole analogues: Determination of their carbonic anhydrase inhibitory activity and molecular modeling studies. | 2019 Jun |
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| 15 |
31072911 | A non-catalytic function of carbonic anhydrase IX contributes to the glycolytic phenotype and pH regulation in human breast cancer cells. | 2019 May 28 |
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| 16 |
31419777 | Carbonic anhydrase inhibitors based on sorafenib scaffold: Design, synthesis, crystallographic investigation and effects on primary breast cancer cells. | 2019 Nov 15 |
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| 17 |
31542715 | Synthesis of coumarin-sulfonamide derivatives and determination of their cytotoxicity, carbonic anhydrase inhibitory and molecular docking studies. | 2019 Dec 1 |
2 |
| 18 |
31810330 | Preclinical Evaluation of Ureidosulfamate Carbonic Anhydrase IX/XII Inhibitors in the Treatment of Cancers. | 2019 Dec 2 |
2 |
| 19 |
29427856 | New anticancer drug candidates sulfonamides as selective hCA IX or hCA XII inhibitors. | 2018 Apr |
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| 20 |
29520697 | The cytotoxic, apoptotic and oxidative effects of carbonic anhydrase IX inhibitor on colorectal cancer cells. | 2018 Apr |
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| 21 |
29571155 | Synthesis of novel 4-functionalized 1,5-diaryl-1,2,3-triazoles containing benzenesulfonamide moiety as carbonic anhydrase I, II, IV and IX inhibitors. | 2018 Apr 25 |
1 |
| 22 |
29778927 | Evaluation of 99mTc-sulfonamide and sulfocoumarin derivatives for imaging carbonic anhydrase IX expression. | 2018 Aug |
1 |
| 23 |
29852328 | Synthesis, characterization and biological evaluation of tertiary sulfonamide derivatives of pyridyl-indole based heteroaryl chalcone as potential carbonic anhydrase IX inhibitors and anticancer agents. | 2018 Jul 15 |
2 |
| 24 |
29965974 | Differential expression and function of CAIX and CAXII in breast cancer: A comparison between tumorgraft models and cells. | 2018 |
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| 25 |
30001631 | Selective inhibition of carbonic anhydrase-IX by sulphonamide derivatives induces pH and reactive oxygen species-mediated apoptosis in cervical cancer HeLa cells. | 2018 Dec |
3 |
| 26 |
30219719 | Tumor-associated carbonic anhydrase isoform IX and XII inhibitory properties of certain isatin-bearing sulfonamides endowed with in vitro antitumor activity towards colon cancer. | 2018 Dec |
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| 27 |
30220229 | Target-based drug discovery through inversion of quantitative structure-drug-property relationships and molecular simulation: CA IX-sulphonamide complexes. | 2018 Dec |
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| 28 |
30452451 | Selective inhibition of carbonic anhydrase IX over carbonic anhydrase XII in breast cancer cells using benzene sulfonamides: Disconnect between activity and growth inhibition. | 2018 |
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| 29 |
30746068 | Novel benzoyl thioureido benzene sulfonamides as highly potent and selective inhibitors of carbonic anhydrase IX: optimization and bioactive studies. | 2018 Dec 1 |
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| 30 |
27774817 | Designing, synthesis and bioactivities of 4-[3-(4-hydroxyphenyl)-5-aryl-4,5-dihydro-pyrazol-1-yl]benzenesulfonamides. | 2017 Dec |
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| 31 |
27890855 | Linker stability influences the anti-tumor activity of acetazolamide-drug conjugates for the therapy of renal cell carcinoma. | 2017 Jan 28 |
2 |
| 32 |
28256371 | Synthesis of bulky-tailed sulfonamides incorporating pyrido[2,3-d][1,2,4]triazolo[4,3-a]pyrimidin-1(5H)-yl) moieties and evaluation of their carbonic anhydrases I, II, IV and IX inhibitory effects. | 2017 Apr 1 |
1 |
| 33 |
28335646 | Synthesis of an acridine orange sulfonamide derivative with potent carbonic anhydrase IX inhibitory action. | 2017 Dec |
1 |
| 34 |
28385087 | Design, synthesis and evaluation of 18F-labeled cationic carbonic anhydrase IX inhibitors for PET imaging. | 2017 Dec |
1 |
| 35 |
28783982 | Quantitative assessment of specific carbonic anhydrase inhibitors effect on hypoxic cells using electrical impedance assays. | 2017 Dec |
1 |
| 36 |
26794023 | Intrinsic thermodynamics of inhibitor binding to human carbonic anhydrase IX. | 2016 Apr |
3 |
| 37 |
27234893 | Synthesis of 4-(thiazol-2-ylamino)-benzenesulfonamides with carbonic anhydrase I, II and IX inhibitory activity and cytotoxic effects against breast cancer cell lines. | 2016 Jul 1 |
2 |
| 38 |
27485269 | Amine coupling versus biotin capture for the assessment of sulfonamide as ligands of hCA isoforms. | 2016 Oct 15 |
1 |
| 39 |
24666294 | Inhibition of human carbonic anhydrase isozymes I, II, IX and XII with a new series of sulfonamides incorporating aroylhydrazone-, [1,2,4]triazolo[3,4-b][1,3,4]thiadiazinyl- or 2-(cyanophenylmethylene)-1,3,4-thiadiazol-3(2H)-yl moieties. | 2015 Feb |
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| 40 |
25875209 | 6-Substituted sulfocoumarins are selective carbonic anhdydrase IX and XII inhibitors with significant cytotoxicity against colorectal cancer cells. | 2015 May 14 |
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| 41 |
25891195 | Designing carbonic anhydrase inhibitors for the treatment of breast cancer. | 2015 Jun |
1 |
| 42 |
26276436 | Carbonic anhydrase inhibitors: Design, synthesis and structural characterization of new heteroaryl-N-carbonylbenzenesulfonamides targeting druggable human carbonic anhydrase isoforms. | 2015 Sep 18 |
1 |
| 43 |
26447758 | Sulfonamide derivative targeting carbonic anhydrase IX as a nuclear imaging probe for colorectal cancer detection in vivo. | 2015 Nov 3 |
4 |
| 44 |
26639945 | Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activity. | 2015 Dec 15 |
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| 45 |
24090422 | Design, synthesis and molecular docking of novel N,N-dimethylbenzenesulfonamide derivatives as potential antiproliferative agents. | 2014 Oct |
2 |
| 46 |
24589511 | Synthesis and carbonic anhydrase I, II, IX and XII inhibition studies of 4-N,N-disubstituted sulfanilamides incorporating 4,4,4-trifluoro-3-oxo-but-1-enyl, phenacylthiourea and imidazol-2(3H)-one/thione moieties. | 2014 Apr 1 |
1 |
| 47 |
24689792 | Cyclic secondary sulfonamides: unusually good inhibitors of cancer-related carbonic anhydrase enzymes. | 2014 Apr 24 |
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| 48 |
25267005 | Inhibition of carbonic anhydrase isoforms I, II, IX and XII with novel Schiff bases: identification of selective inhibitors for the tumor-associated isoforms over the cytosolic ones. | 2014 Nov 1 |
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| 49 |
25358036 | A class of 4-sulfamoylphenyl-ω-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects. | 2014 Nov 26 |
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| 50 |
23168081 | New selective carbonic anhydrase IX inhibitors: synthesis and pharmacological evaluation of diarylpyrazole-benzenesulfonamides. | 2013 Mar 15 |
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