Cocaine

solute carrier family 6 member 4 ; Homo sapiens







73 Article(s)
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1 34798166 Methylation of the serotonin transporter gene moderates the depressive subjective effect of cocaine. 2022 Feb 10 7
2 33658787 Association of Serotonin Transporter (SERT) Polymorphisms with Opioid Dependence and Dimensional Aspects of Cocaine Use in a Caucasian Cohort of Opioid Users. 2021 6
3 33785354 Functional characterization of N-octyl 4-methylamphetamine variants and related bivalent compounds at the dopamine and serotonin transporters using Ca2+ channels as sensors. 2021 May 15 1
4 33888022 An efficient and label-free LC-MS/MS method for assessing drug's activity at dopamine and serotonin transporters using transporter-transfected HEK293T cells. 2021 Jun 1
5 34199621 Functional Characterization of the Dopaminergic Psychostimulant Sydnocarb as an Allosteric Modulator of the Human Dopamine Transporter. 2021 Jun 2 1
6 32494974 Serotonin transporter protein in autopsied brain of chronic users of cocaine. 2020 Sep 16
7 30680295 Detection of Ligand-binding to Membrane Proteins by Capacitance Measurements. 2019 Jan 5 2
8 31570504 Serotonin transport in the 21st century. 2019 Nov 4 1
9 29357981 Median and Dorsal Raphe Serotonergic Neurons Control Moderate Versus Compulsive Cocaine Intake. 2018 Jun 15 2
10 28590957 Genetic moderation of cocaine subjective effects by variation in the TPH1, TPH2, and SLC6A4 serotonin genes. 2017 Oct 4
11 27140629 Control of serotonin transporter phosphorylation by conformational state. 2016 May 17 1
12 25873594 Ligand Selectivity among the Dopamine and Serotonin Transporters Specified by the Forward Binding Reaction. 2015 Jul 3
13 26110342 Serotonin transporter gene promoter polymorphism predicts relationship between years of cocaine use and impulsivity. 2015 Oct 1
14 24081522 Extracellular loop 3 of the noradrenaline transporter contributes to substrate and inhibitor selectivity. 2014 Jan 1
15 24973209 The serotonin transporter undergoes constitutive internalization and is primarily sorted to late endosomes and lysosomal degradation. 2014 Aug 15 1
16 23518607 Multi-cultural association of the serotonin transporter gene (SLC6A4) with substance use disorder. 2013 Aug 2
17 23706649 Thermostabilisation of the serotonin transporter in a cocaine-bound conformation. 2013 Jun 26 2
18 23776432 Ligand induced conformational changes of the human serotonin transporter revealed by molecular dynamics simulations. 2013 1
19 24120036 Lack of association between the LPR and VNTR polymorphisms of the serotonin transporter gene and cocaine dependence in a Spanish sample. 2013 Dec 30 1
20 21309950 The SLC6A4 VNTR genotype determines transcription factor binding and epigenetic variation of this gene in response to cocaine in vitro. 2012 Jan 3
21 22925276 Modifying the role of serotonergic 5-HTTLPR and TPH2 variants on disulfiram treatment of cocaine addiction: a preliminary study. 2012 Nov 1
22 20932493 Drugs of abuse and human placenta. 2011 May 23 1
23 21146984 The synthesis and biological evaluation of 2-(3-methyl or 3-phenylisoxazol-5-yl)-3-aryl-8-thiabicyclo[3.2.1]octanes. 2011 Jan 1 2
24 21420984 Interaction of tyrosine 151 in norepinephrine transporter with the 2β group of cocaine analog RTI-113. 2011 Jul-Aug 1
25 22379462 Prenatal Cocaine Disrupts Serotonin Signaling-Dependent Behaviors: Implications for Sex Differences, Early Stress and Prenatal SSRI Exposure. 2011 Sep 2
26 20159976 Transmembrane domain 6 of the human serotonin transporter contributes to an aqueously accessible binding pocket for serotonin and the psychostimulant 3,4-methylene dioxymethamphetamine. 2010 Apr 9 2
27 19351213 Development and validation of a high-throughput screening method for two polymorphisms in the serotonin transporter gene. 2009 1
28 19572987 Upregulation of serotonin transporter by alcohol in human dendritic cells: possible implication in neuroimmune deregulation. 2009 Oct 1
29 19837674 Ligand effects on cross-linking support a conformational mechanism for serotonin transport. 2009 Dec 4 1
30 18321529 Relationship of the serotonin transporter with prolactin response to meta-chlorophenylpiperazine in cocaine dependence. 2008 Oct 3
31 19075665 Computational approaches for the study of serotonin and its membrane transporter SERT: implications for drug design in neurological sciences. 2008 1
32 19086766 Nonhuman primate neuroimaging and cocaine medication development. 2008 Dec 4
33 17698848 Ibogaine, a noncompetitive inhibitor of serotonin transport, acts by stabilizing the cytoplasm-facing state of the transporter. 2007 Oct 5 1
34 16272152 Tyr-95 and Ile-172 in transmembrane segments 1 and 3 of human serotonin transporters interact to establish high affinity recognition of antidepressants. 2006 Jan 27 1
35 16451060 Evaluation of carbon-11-labeled 2beta-carbomethoxy-3beta-[4'-((Z)-2-iodoethenyl)phenyl]nortropane as a potential radioligand for imaging the serotonin transporter by PET. 2006 Feb 9 3
36 16515684 Comparison of the monoamine transporters from human and mouse in their sensitivities to psychostimulant drugs. 2006 Mar 3 3
37 17000009 Polymorphism in the serotonin transporter gene and moderators of prolactin response to meta-chlorophenylpiperazine in African-American cocaine abusers and controls. 2006 Nov 15 1
38 16109588 Polymorphism in the serotonin transporter gene and response to treatment in African American cocaine and alcohol-abusing individuals. 2005 Sep 2
39 16112691 Serotonin transporter mutations associated with obsessive-compulsive disorder and phosphorylation alter binding affinity for inhibitors. 2005 Nov 1
40 16250852 PET and SPECT exploration of central monoaminergic transporters for the development of new drugs and treatments in brain disorders. 2005 1
41 14593087 Distinct molecular recognition of psychostimulants by human and Drosophila serotonin transporters. 2004 Feb 1
42 15091312 Relationship between serotonin transporter gene polymorphisms and platelet serotonin transporter sites among African-American cocaine-dependent individuals and healthy volunteers. 2004 Mar 4
43 21473026 2β-Carbo[11C]methoxy-3β-(4´-((Z)-2-iodoethenyl)phenyl)nortropane 2004 1
44 12590403 Seasonal variations in the binding of [3H]paroxetine to the platelet serotonin transporter sites in African-American cocaine-dependent patients and healthy volunteers. 2003 Mar 1
45 14644011 Plasticity in serotonin control mechanisms in the gut. 2003 Dec 1
46 11904159 Voltage-dependent transient currents of human and rat 5-HT transporters (SERT) are blocked by HEPES and ion channel ligands. 2002 Feb 27 1
47 12057823 Serotonin transporter polymorphisms and measures of impulsivity, aggression, and sensation seeking among African-American cocaine-dependent individuals. 2002 Jun 1 4
48 12180970 A cocaine insensitive chimeric insect serotonin transporter reveals domains critical for cocaine interaction. 2002 Aug 5
49 12218660 No association between polymorphisms in the serotonin transporter gene and susceptibility to cocaine dependence among African-American individuals. 2002 Sep 2
50 12491807 [Pharmacology of monoamine neurotransmitter transporters]. 2002 Nov 1