Terfenadine

potassium voltage-gated channel subfamily H member 2 ; Homo sapiens







16 Article(s)
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1 31664867 Investigating the utility of adult zebrafish ex vivo whole hearts to pharmacologically screen hERG channel activator compounds. 2019 Dec 1 1
2 26376488 Molecular Cloning and Functional Expression of the Equine K+ Channel KV11.1 (Ether à Go-Go-Related/KCNH2 Gene) and the Regulatory Subunit KCNE2 from Equine Myocardium. 2015 1
3 25366487 Effect of terfenadine and pentamidine on the HERG channel and its intracellular trafficking: combined analysis with automated voltage clamp and confocal microscopy. 2014 1
4 23221912 Role of the activation gate in determining the extracellular potassium dependency of block of HERG by trapped drugs. 2013 Jan 1 2
5 14709917 Lack of action potential-prolonging effect of terfenadine on rabbit myocardial tissue preparations. 2004 Jan 1
6 15272206 Validation of a [3H]astemizole binding assay in HEK293 cells expressing HERG K+ channels. 2004 Jul 1
7 11575008 [The effect of second generation histamine antagonists on the heart]. 2001 1
8 10604956 Loratadine blockade of K(+) channels in human heart: comparison with terfenadine under physiological conditions. 2000 Jan 1
9 10828461 Redox state dependency of HERGS631C channel pharmacology: relation to C-type inactivation. 2000 May 26 1
10 10422790 Epinastine, a nonsedating histamine H1 receptor antagonist, has a negligible effect on HERG channel. 1999 Jun 25 2
11 10444235 Cardiac ion channels and antihistamines: possible mechanisms of cardiotoxicity. 1999 Jul 1
12 9658196 Molecular basis for the lack of HERG K+ channel block-related cardiotoxicity by the H1 receptor blocker cetirizine compared with other second-generation antihistamines. 1998 Jul 2
13 9694927 Blockade of HERG and Kv1.5 by ketoconazole. 1998 Aug 3
14 9714291 Human ether-a-gogo related gene (HERG) K+ channels as pharmacological targets: present and future implications. 1998 Jun 1 1
15 8641472 Blockade of HERG channels expressed in Xenopus oocytes by the histamine receptor antagonists terfenadine and astemizole. 1996 Apr 29 3
16 8772706 HERG, a primary human ventricular target of the nonsedating antihistamine terfenadine. 1996 Aug 15 3