12 Article(s)Download |
PMID | Title | Pub. Year | #Total Relationships |
1 | 31303995 | Discovery of (aza)indole derivatives as novel respiratory syncytial virus fusion inhibitors. | 2019 Jun 1 | 1 |
2 | 23681056 | Virtual screening and structure-based discovery of indole acylguanidines as potent β-secretase (BACE1) inhibitors. | 2013 May 16 | 1 |
3 | 22104146 | II. Novel HCV NS5B polymerase inhibitors: discovery of indole C2 acyl sulfonamides. | 2012 Jan 1 | 1 |
4 | 22607682 | Sulfonyl-morpholino-pyrimidines: SAR and development of a novel class of selective mTOR kinase inhibitor. | 2012 Jun 15 | 1 |
5 | 19914828 | 5-Lipoxygenase-activating protein inhibitors. Part 2: 3-{5-((S)-1-Acetyl-2,3-dihydro-1H-indol-2-ylmethoxy)-3-tert-butylsulfanyl-1-[4-(5-methoxy-pyrimidin-2-yl)-benzyl]-1H-indol-2-yl}-2,2-dimethyl-propionic acid (AM679)--a potent FLAP inhibitor. | 2010 Jan 1 | 2 |
6 | 20074949 | N-Acetamideindolecarboxylic acid allosteric 'finger-loop' inhibitors of the hepatitis C virus NS5B polymerase: discovery and initial optimization studies. | 2010 Feb 1 | 1 |
7 | 19769332 | Inhibitors of human immunodeficiency virus type 1 (HIV-1) attachment. 5. An evolution from indole to azaindoles leading to the discovery of 1-(4-benzoylpiperazin-1-yl)-2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione (BMS-488043), a drug candidate that demonstrates antiviral activity in HIV-1-infected subjects. | 2009 Dec 10 | 1 |
8 | 18308566 | Indole- and indolizine-glyoxylamides displaying cytotoxicity against multidrug resistant cancer cell lines. | 2008 Mar 15 | 1 |
9 | 17512197 | Synthesis and SAR of selective benzothiophene, benzofuran, and indole-based peroxisome proliferator-activated receptor delta agonists. | 2007 Jul 1 | 2 |
10 | 15186849 | Discovery and SAR of indole-2-carboxylic acid benzylidene-hydrazides as a new series of potent apoptosis inducers using a cell-based HTS assay. | 2004 Jul 1 | 1 |
11 | 15546707 | Tryptamine-based human beta3-adrenergic receptor agonists. Part 1: SAR studies of the 7-position of the indole ring. | 2004 Dec 20 | 1 |
12 | 12729661 | Non-imidazole heterocyclic histamine H3 receptor antagonists. | 2003 May 19 | 1 |