indole

sarcosine dehydrogenase ; Homo sapiens







12 Article(s)
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Pub. Year
#Total Relationships
1 31303995 Discovery of (aza)indole derivatives as novel respiratory syncytial virus fusion inhibitors. 2019 Jun 1 1
2 23681056 Virtual screening and structure-based discovery of indole acylguanidines as potent β-secretase (BACE1) inhibitors. 2013 May 16 1
3 22104146 II. Novel HCV NS5B polymerase inhibitors: discovery of indole C2 acyl sulfonamides. 2012 Jan 1 1
4 22607682 Sulfonyl-morpholino-pyrimidines: SAR and development of a novel class of selective mTOR kinase inhibitor. 2012 Jun 15 1
5 19914828 5-Lipoxygenase-activating protein inhibitors. Part 2: 3-{5-((S)-1-Acetyl-2,3-dihydro-1H-indol-2-ylmethoxy)-3-tert-butylsulfanyl-1-[4-(5-methoxy-pyrimidin-2-yl)-benzyl]-1H-indol-2-yl}-2,2-dimethyl-propionic acid (AM679)--a potent FLAP inhibitor. 2010 Jan 1 2
6 20074949 N-Acetamideindolecarboxylic acid allosteric 'finger-loop' inhibitors of the hepatitis C virus NS5B polymerase: discovery and initial optimization studies. 2010 Feb 1 1
7 19769332 Inhibitors of human immunodeficiency virus type 1 (HIV-1) attachment. 5. An evolution from indole to azaindoles leading to the discovery of 1-(4-benzoylpiperazin-1-yl)-2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione (BMS-488043), a drug candidate that demonstrates antiviral activity in HIV-1-infected subjects. 2009 Dec 10 1
8 18308566 Indole- and indolizine-glyoxylamides displaying cytotoxicity against multidrug resistant cancer cell lines. 2008 Mar 15 1
9 17512197 Synthesis and SAR of selective benzothiophene, benzofuran, and indole-based peroxisome proliferator-activated receptor delta agonists. 2007 Jul 1 2
10 15186849 Discovery and SAR of indole-2-carboxylic acid benzylidene-hydrazides as a new series of potent apoptosis inducers using a cell-based HTS assay. 2004 Jul 1 1
11 15546707 Tryptamine-based human beta3-adrenergic receptor agonists. Part 1: SAR studies of the 7-position of the indole ring. 2004 Dec 20 1
12 12729661 Non-imidazole heterocyclic histamine H3 receptor antagonists. 2003 May 19 1