| 1 |
34323202 | An Update of Lysine Specific Demethylase 1 Inhibitor: A Patent Review (2016-2020). | 2022 |
2 |
| 2 |
34718134 | Therapeutic potential of targeting LSD1/ KDM1A in cancers. | 2022 Jan |
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| 3 |
33527838 | Raloxifene, identified as a novel LSD1 inhibitor, suppresses the migration of renal cell carcinoma. | 2021 Mar |
2 |
| 4 |
33729758 | Design, Synthesis, and Evaluation of (2-Aminocyclopropyl)phenyl Derivatives as Novel Positron Emission Tomography Imaging Agents for Lysine-Specific Demethylase 1 in the Brain. | 2021 Apr 8 |
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| 5 |
34423983 | Design, Synthesis, and Evaluation of [18F]T-914 as a Novel Positron-Emission Tomography Tracer for Lysine-Specific Demethylase 1. | 2021 Sep 9 |
4 |
| 6 |
32166890 | Development and Structural Evaluation of N-Alkylated trans-2-Phenylcyclopropylamine-Based LSD1 Inhibitors. | 2020 May 6 |
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| 7 |
33088686 | Exploration of 5-cyano-6-phenylpyrimidin derivatives containing an 1,2,3-triazole moiety as potent FAD-based LSD1 inhibitors. | 2020 Sep |
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| 8 |
29198865 | Histone H3 peptides incorporating modified lysine residues as lysine-specific demethylase 1 inhibitors. | 2018 Jan 15 |
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| 9 |
29247860 | Structure-activity studies on N-Substituted tranylcypromine derivatives lead to selective inhibitors of lysine specific demethylase 1 (LSD1) and potent inducers of leukemic cell differentiation. | 2018 Jan 20 |
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| 10 |
29921310 | KDM1A microenvironment, its oncogenic potential, and therapeutic significance. | 2018 Jun 19 |
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| 11 |
28279976 | Regulation of hypoxia responses by flavin adenine dinucleotide-dependent modulation of HIF-1α protein stability. | 2017 Apr 13 |
4 |
| 12 |
29088714 | Inhibition of LSD1 epigenetically attenuates oral cancer growth and metastasis. | 2017 Sep 26 |
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| 13 |
29156705 | Upregulation of CD11b and CD86 through LSD1 inhibition promotes myeloid differentiation and suppresses cell proliferation in human monocytic leukemia cells. | 2017 Oct 17 |
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| 14 |
26673564 | Lysine-Specific Demethylase 1A (KDM1A/LSD1): Product Recognition and Kinetic Analysis of Full-Length Histones. | 2016 Mar 22 |
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| 15 |
27059868 | Inhibition of Lysine-Specific Demethylase-1 (LSD1/KDM1A) Promotes the Adipogenic Differentiation of hESCs Through H3K4 Methylation. | 2016 Jun |
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| 16 |
27634040 | Activity-dependent Regulation of Histone Lysine Demethylase KDM1A by a Putative Thiol/Disulfide Switch. | 2016 Nov 18 |
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| 17 |
25827878 | In vitro histone demethylase assays. | 2015 |
4 |
| 18 |
26230878 | Hologram quantitative structure-activity relationship and comparative molecular interaction field analysis of aminothiazole and thiazolesulfonamide as reversible LSD1 inhibitors. | 2015 |
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| 19 |
25103574 | Low activity of LSD1 elicits a pro-inflammatory gene expression profile in riboflavin-deficient human T Lymphoma Jurkat cells. | 2014 Sep |
4 |
| 20 |
23988016 | Amine oxidation mediated by lysine-specific demethylase 1: quantum mechanics/molecular mechanics insights into mechanism and role of lysine 661. | 2013 Sep 11 |
4 |
| 21 |
22132744 | Oligoamine analogues in combination with 2-difluoromethylornithine synergistically induce re-expression of aberrantly silenced tumour-suppressor genes. | 2012 Mar 15 |
1 |
| 22 |
22339659 | Lysine-specific histone demethylase 1 (LSD1): A potential molecular target for tumor therapy. | 2012 |
4 |
| 23 |
20970991 | Structural insights into histone lysine demethylation. | 2010 Dec |
4 |
| 24 |
19381934 | In vitro histone demethylase assays. | 2009 |
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| 25 |
19624733 | New roles of flavoproteins in molecular cell biology: histone demethylase LSD1 and chromatin. | 2009 Aug |
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| 26 |
18039463 | Crystal structure of histone demethylase LSD1 and tranylcypromine at 2.25 A. | 2008 Feb 1 |
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| 27 |
17529991 | Structural basis of histone demethylation by LSD1 revealed by suicide inactivation. | 2007 Jun |
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| 28 |
17569509 | Structural basis for the inhibition of the LSD1 histone demethylase by the antidepressant trans-2-phenylcyclopropylamine. | 2007 Jul 10 |
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| 29 |
17101443 | Purification of histone demethylases from HeLa cells. | 2006 Dec |
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