| 1 |
34710811 | Atomistic insights into the selective therapeutic activity of 6-(2,4-difluorophenoxy)-5-((ethylmethyl)pyridine-3-yl)-8-methylpyrrolo[1,2-a]pyrazin-1(2H)-one towards bromodomain-containing proteins. | 2021 Dec |
1 |
| 2 |
34845959 | Theoretically exploring selective-binding mechanisms of BRD4 through integrative computational approaches. | 2021 Dec |
1 |
| 3 |
32657160 | Probing molecular mechanism of inhibitor bindings to bromodomain-containing protein 4 based on molecular dynamics simulations and principal component analysis. | 2020 Jul |
1 |
| 4 |
31857841 | Evaluating the Advantages of Using 3D-Enriched Fragments for Targeting BET Bromodomains. | 2019 Dec 12 |
1 |
| 5 |
28983974 | Molecular design of Stat3-derived peptide selectivity between BET proteins Brd2 and Brd4 in ovarian cancer. | 2018 Feb |
1 |
| 6 |
29649741 | Discovery of potent and selective BRD4 inhibitors capable of blocking TLR3-induced acute airway inflammation. | 2018 May 10 |
1 |
| 7 |
29776834 | BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability. | 2018 Jul 15 |
1 |
| 8 |
30411639 | In silico study directed towards identification of novel high-affinity inhibitors targeting an oncogenic protein: BRD4-BD1. | 2018 Dec |
2 |
| 9 |
26191363 | BRD4 Structure-Activity Relationships of Dual PLK1 Kinase/BRD4 Bromodomain Inhibitor BI-2536. | 2015 Jul 9 |
1 |
| 10 |
24767840 | Discovery of BRD4 bromodomain inhibitors by fragment-based high-throughput docking. | 2014 Jun 1 |
1 |