BI 2536

bromodomain containing 4 ; Homo sapiens







5 Article(s)
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#Total Relationships
1 33638254 Design, synthesis, and biological evaluation of novel 4,4-difluoro-1-methyl-N, 6-diphenyl-5, 6-dihydro-4H-pyrimido [4, 5-b] [1, 2, 4] triazolo [4, 3-d] [1, 4] diazepin-8-amine derivatives as potential BRD4 inhibitors. 2021 May 1
2 29525435 Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups. 2018 Apr 25 2
3 28586718 Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor. 2017 Sep 8 1
4 26191363 BRD4 Structure-Activity Relationships of Dual PLK1 Kinase/BRD4 Bromodomain Inhibitor BI-2536. 2015 Jul 9 5
5 24568369 Acetyl-lysine binding site of bromodomain-containing protein 4 (BRD4) interacts with diverse kinase inhibitors. 2014 May 16 1