| 1 |
34596922 | Novel benzenesulfonamide-bearing pyrazoles and 1,2,4-thiadiazoles as selective carbonic anhydrase inhibitors. | 2022 Jan |
1 |
| 2 |
33249154 | Utilization of the common functional groups in bioactive molecules: Exploring dual inhibitory potential and computational analysis of keto esters against α-glucosidase and carbonic anhydrase-II enzymes. | 2021 Jan 15 |
1 |
| 3 |
34387019 | Inhibition Profiles of Some Symmetric Sulfamides Derived from Phenethylamines on Human Carbonic Anhydrase I, and II Isoenzymes. | 2021 Oct |
1 |
| 4 |
31911296 | Structure-activity relationship of human carbonic anhydrase-II inhibitors: Detailed insight for future development as anti-glaucoma agents. | 2020 Jan |
1 |
| 5 |
33085484 | Structural Basis of Nanomolar Inhibition of Tumor-Associated Carbonic Anhydrase IX: X-Ray Crystallographic and Inhibition Study of Lipophilic Inhibitors with Acetazolamide Backbone. | 2020 Nov 12 |
1 |
| 6 |
30535510 | Repeatability, precision, and accuracy of the enthalpies and Gibbs energies of a protein-ligand binding reaction measured by isothermal titration calorimetry. | 2019 Mar |
5 |
| 7 |
30597695 | Evaluation of antimicrobial, antibiofilm and carbonic anhydrase inhibition profiles of 1,3-bis-chalcone derivatives. | 2019 Apr |
1 |
| 8 |
31345748 | Sulfonate and sulfamate derivatives possessing benzofuran or benzothiophene nucleus as potent carbonic anhydrase II/IX/XII inhibitors. | 2019 Sep 1 |
1 |
| 9 |
31555842 | Obtaining precise and accurate results by ITC. | 2019 Dec |
1 |
| 10 |
31667562 | Automated and enhanced extraction of a small molecule-drug conjugate using an enzyme-inhibitor interaction based SPME tool followed by direct analysis by ESI-MS. | 2019 Nov |
2 |
| 11 |
31847904 | Carbonic anhydrase 2 (CAII) supports tumor blood endothelial cell survival under lactic acidosis in the tumor microenvironment. | 2019 Dec 17 |
1 |
| 12 |
28792233 | Synthesis of chalcone-imide derivatives and investigation of their anticancer and antimicrobial activities, carbonic anhydrase and acetylcholinesterase enzymes inhibition profiles. | 2018 Feb |
1 |
| 13 |
29149534 | Novel N-propylphthalimide- and 4-vinylbenzyl-substituted benzimidazole salts: Synthesis, characterization, and determination of their metal chelating effects and inhibition profiles against acetylcholinesterase and carbonic anhydrase enzymes. | 2018 Jan |
1 |
| 14 |
29197732 | Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases. | 2018 Jan 1 |
2 |
| 15 |
29283199 | Synthesis and investigation of the conversion reactions of pyrimidine-thiones with nucleophilic reagent and evaluation of their acetylcholinesterase, carbonic anhydrase inhibition, and antioxidant activities. | 2018 Feb |
1 |
| 16 |
29584404 | Dual-Valve and Counter-Flow Surface Plasmon Resonance. | 2018 Apr 17 |
1 |
| 17 |
30153589 | Novel sulfonamides incorporating 1,3,5-triazine and amino acid structural motifs as inhibitors of the physiological carbonic anhydrase isozymes I, II and IV and tumor-associated isozyme IX. | 2018 Dec |
1 |
| 18 |
27780313 | Synthesis, carbonic anhydrase I and II isoenzymes inhibition properties, and antibacterial activities of novel tetralone-based 1,4-benzothiazepine derivatives. | 2017 Apr |
1 |
| 19 |
27984137 | Novel eugenol derivatives: Potent acetylcholinesterase and carbonic anhydrase inhibitors. | 2017 Jan |
1 |
| 20 |
28100082 | Synthesis and bioactivity of several new hetaryl sulfonamides. | 2017 Dec |
1 |
| 21 |
28110167 | Chiral separation of new sulfonamide derivatives and evaluation of their enantioselective affinity for human carbonic anhydrase II by microscale thermophoresis and surface plasmon resonance. | 2017 Apr 15 |
1 |
| 22 |
28117934 | Synthesis of new cyclic thioureas and evaluation of their metal-chelating activity, acetylcholinesterase, butyrylcholinesterase, and carbonic anhydrase inhibition profiles. | 2017 Jul |
2 |
| 23 |
28544359 | Discovery of potent carbonic anhydrase, acetylcholinesterase, and butyrylcholinesterase enzymes inhibitors: The new amides and thiazolidine-4-ones synthesized on an acetophenone base. | 2017 Sep |
1 |
| 24 |
28943245 | Improved molecular recognition of Carbonic Anhydrase IX by polypeptide conjugation to acetazolamide. | 2017 Oct 15 |
2 |
| 25 |
26985691 | Synthesis and inhibitory properties of some carbamates on carbonic anhydrase and acetylcholine esterase. | 2016 Dec |
1 |
| 26 |
27050248 | Synthesis of some tetrahydropyrimidine-5-carboxylates, determination of their metal chelating effects and inhibition profiles against acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase. | 2016 Dec |
1 |
| 27 |
27075164 | The synthesis of some β-lactams and investigation of their metal-chelating activity, carbonic anhydrase and acetylcholinesterase inhibition profiles. | 2016 |
1 |
| 28 |
27232456 | Molecular dynamics study of human carbonic anhydrase II in complex with Zn(2+) and acetazolamide on the basis of all-atom force field simulations. | 2016 Jul-Aug |
2 |
| 29 |
27579806 | Synthesis, cytotoxicity and carbonic anhydrase inhibitory activities of new pyrazolines. | 2016 |
1 |
| 30 |
27717855 | Isothermal titration calorimetry for drug design: Precision of the enthalpy and binding constant measurements and comparison of the instruments. | 2016 Dec 15 |
1 |
| 31 |
28461893 | Neutron structure of human carbonic anhydrase II in complex with methazolamide: mapping the solvent and hydrogen-bonding patterns of an effective clinical drug. | 2016 Sep 1 |
2 |
| 32 |
25581127 | Carbonic anhydrase inhibitors with dual-tail moieties to match the hydrophobic and hydrophilic halves of the carbonic anhydrase active site. | 2015 Feb 12 |
1 |
| 33 |
26041446 | Carbonic anhydrase II binds to and increases the activity of the epithelial sodium-proton exchanger, NHE3. | 2015 Aug 15 |
1 |
| 34 |
26105196 | Sulfonamide bearing pyrazolylpyrazolines as potent inhibitors of carbonic anhydrase isoforms I, II, IX and XII. | 2015 Aug 15 |
1 |
| 35 |
24682061 | New aromatic/heteroaromatic propanesulfonylhydrazone compounds: synthesis, physical properties and inhibition studies against carbonic anhydrase II (CAII) enzyme. | 2014 Jul 15 |
1 |
| 36 |
25456084 | 4-Functionalized 1,3-diarylpyrazoles bearing 6-aminosulfonylbenzothiazole moiety as potent inhibitors of carbonic anhydrase isoforms hCA I, II, IX and XII. | 2014 Dec 15 |
1 |
| 37 |
22145674 | Inhibition of mammalian carbonic anhydrase isoforms I, II and VI with thiamine and thiamine-like molecules. | 2013 Apr |
1 |
| 38 |
23633596 | Effects of cryoprotectants on the structure and thermostability of the human carbonic anhydrase II-acetazolamide complex. | 2013 May |
6 |
| 39 |
22928733 | Neutron diffraction of acetazolamide-bound human carbonic anhydrase II reveals atomic details of drug binding. | 2012 Sep 12 |
1 |
| 40 |
19231207 | Carbonic anhydrase inhibitors. Inhibition of human erythrocyte isozymes I and II with a series of antioxidant phenols. | 2009 Apr 15 |
1 |
| 41 |
19851004 | High-resolution structure of human carbonic anhydrase II complexed with acetazolamide reveals insights into inhibitor drug design. | 2009 Oct 1 |
6 |
| 42 |
18295485 | Carbonic anhydrase inhibitors: the very weak inhibitors dithiothreitol, beta-mercaptoethanol, tris(carboxyethyl)phosphine and threitol interfere with the binding of sulfonamides to isozymes II and IX. | 2008 Mar 15 |
1 |
| 43 |
17614791 | Reconstitution of carbonic anhydrase activity of the cell-surface-binding protein of vaccinia virus. | 2007 Oct 1 |
1 |
| 44 |
15110853 | Carbonic anhydrase inhibitors: aromatic and heterocyclic sulfonamides incorporating adamantyl moieties with strong anticonvulsant activity. | 2004 May 15 |
1 |
| 45 |
15183767 | Comparative analyses of a small molecule/enzyme interaction by multiple users of Biacore technology. | 2004 Jul 1 |
2 |
| 46 |
12767917 | Inhibition of carbonic anhydrase II by steroidal and non-steroidal sulphamates. | 2003 Jun 13 |
1 |
| 47 |
14611844 | Carbonic anhydrase inhibitors: inhibition of human and murine mitochondrial isozymes V with anions. | 2003 Sep 1 |
1 |
| 48 |
12027220 | Na+:HCO3- cotransporters (NBC): expression and regulation in the kidney. | 2002 Mar-Apr |
2 |
| 49 |
12138085 | Carbonic anhydrase II binds to and enhances activity of the Na+/H+ exchanger. | 2002 Sep 27 |
1 |
| 50 |
12372813 | The functional and physical relationship between the DRA bicarbonate transporter and carbonic anhydrase II. | 2002 Nov |
1 |