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23316861 | Preclinical evaluation of carbon-11 and fluorine-18 sulfonamide derivatives for in vivo radiolabeling of erythrocytes. | 2013 Jan 15 |
2 |
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23352754 | o-Benzenedisulfonimido-sulfonamides are potent inhibitors of the tumor-associated carbonic anhydrase isoforms CA IX and CA XII. | 2013 Mar 15 |
1 |
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23777898 | Sulfonamides containing coumarin moieties selectively and potently inhibit carbonic anhydrases II and IX: design, synthesis, inhibitory activity and 3D-QSAR analysis. | 2013 Aug |
1 |
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23859774 | 5-Substituted-(1,2,3-triazol-4-yl)thiophene-2-sulfonamides strongly inhibit human carbonic anhydrases I, II, IX and XII: solution and X-ray crystallographic studies. | 2013 Sep 1 |
2 |
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24012377 | Structural study of the location of the phenyl tail of benzene sulfonamides and the effect on human carbonic anhydrase inhibition. | 2013 Nov 1 |
1 |
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22386980 | Mutation of active site residues Asn67 to Ile, Gln92 to Val and Leu204 to Ser in human carbonic anhydrase II: influences on the catalytic activity and affinity for inhibitors. | 2012 Apr 1 |
1 |
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22775345 | Development of potent carbonic anhydrase inhibitors incorporating both sulfonamide and sulfamide groups. | 2012 Aug 9 |
1 |
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21371595 | Protein thermal shifts to identify low molecular weight fragments. | 2011 |
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21706094 | Human carbonic anhydrase II as a host for piano-stool complexes bearing a sulfonamide anchor. | 2011 Aug 7 |
1 |
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20005709 | Carbonic anhydrase inhibitors. X-ray crystal studies of the carbonic anhydrase II-trithiocarbonate adduct--an inhibitor mimicking the sulfonamide and urea binding to the enzyme. | 2010 Jan 15 |
1 |
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20371220 | Kinetic analysis and fragment screening with Fujifilm AP-3000. | 2010 Jul 15 |
1 |
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20598552 | Coumarinyl-substituted sulfonamides strongly inhibit several human carbonic anhydrase isoforms: solution and crystallographic investigations. | 2010 Jul 15 |
2 |
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20819062 | 3-phenyl-1H-indole-5-sulfonamides: structure-based drug design of a promising class of carbonic anhydrase inhibitors. | 2010 |
1 |
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19201197 | Carbonic anhydrase inhibitors. The nematode alpha-carbonic anhydrase of Caenorhabditis elegans CAH-4b is highly inhibited by 2-(hydrazinocarbonyl)-3-substituted-phenyl-1H-indole-5-sulfonamides. | 2009 Apr 15 |
1 |
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19231207 | Carbonic anhydrase inhibitors. Inhibition of human erythrocyte isozymes I and II with a series of antioxidant phenols. | 2009 Apr 15 |
1 |
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19303173 | A QSAR study on relationship between structure of sulfonamides and their carbonic anhydrase inhibitory activity using the eigenvalue (EVA) method. | 2009 Sep |
1 |
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19778001 | Dissecting the inhibition mechanism of cytosolic versus transmembrane carbonic anhydrases by ESR. | 2009 Oct 22 |
2 |
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19796939 | Carbonic anhydrase II-induced selection of inhibitors from a dynamic combinatorial library of Schiff's bases. | 2009 Nov 1 |
1 |
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19824891 | Carbonic anhydrase inhibitors: glycosylsulfanilamides act as subnanomolar inhibitors of the human secreted isoform VI. | 2009 Dec |
1 |
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19827837 | S-glycosyl primary sulfonamides--a new structural class for selective inhibition of cancer-associated carbonic anhydrases. | 2009 Oct 22 |
1 |
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18037297 | Properties of flaky affinity resin with co-continuous structure. | 2008 Feb 15 |
1 |
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18162396 | Carbonic anhydrase inhibitors. Interaction of 2-N,N-dimethylamino-1,3,4-thiadiazole-5-methanesulfonamide with 12 mammalian isoforms: kinetic and X-ray crystallographic studies. | 2008 Feb 1 |
1 |
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18179217 | Using ion channel-forming peptides to quantify protein-ligand interactions. | 2008 Jan 30 |
3 |
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18599640 | A quantitative model of thermal stabilization and destabilization of proteins by ligands. | 2008 Oct |
1 |
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18600270 | Carbonic anhydrase inhibitors. Sulfonamide diuretics revisited--old leads for new applications? | 2008 Jul 21 |
2 |
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17118494 | 3D-QSAR study of sulfonamide inhibitors of human carbonic anhydrase II. | 2007 Mar |
3 |
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17504133 | Dual carbonic anhydrase--cyclooxygenase-2 inhibitors. | 2007 |
1 |
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16787097 | Carbonic anhydrase inhibitors: X-ray and molecular modeling study for the interaction of a fluorescent antitumor sulfonamide with isozyme II and IX. | 2006 Jun 28 |
1 |
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16820676 | X-ray crystallographic studies reveal that the incorporation of spacer groups in carbonic anhydrase inhibitors causes alternate binding modes. | 2006 Jul 1 |
1 |
| 80 |
16858005 | Inhibition profiling of human carbonic anhydrase II by high-throughput screening of structurally diverse, biologically active compounds. | 2006 Oct |
1 |
| 81 |
16962556 | Exploring "one-shot" kinetics and small molecule analysis using the ProteOn XPR36 array biosensor. | 2006 Nov 15 |
1 |
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17007806 | Comparative analysis of 10 small molecules binding to carbonic anhydrase II by different investigators using Biacore technology. | 2006 Dec 1 |
1 |
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15603956 | Carbonic anhydrase inhibitors. Novel sulfanilamide/acetazolamide derivatives obtained by the tail approach and their interaction with the cytosolic isozymes I and II, and the tumor-associated isozyme IX. | 2005 Jan 17 |
1 |
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15686888 | QSAR studies on benzene sulfonamide carbonic anhydrase inhibitors: need of hydrophobic parameter for topological modeling of binding constants of sulfonamides to human CA-II. | 2005 Feb 15 |
2 |
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16134940 | Carbonic anhydrase inhibitors: stacking with Phe131 determines active site binding region of inhibitors as exemplified by the X-ray crystal structure of a membrane-impermeant antitumor sulfonamide complexed with isozyme II. | 2005 Sep 8 |
1 |
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16165351 | Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with benzo[b]thiophene 1,1-dioxide sulfonamides. | 2005 Nov 1 |
1 |
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16298304 | The binding of human carbonic anhydrase II by functionalized folded polypeptide receptors. | 2005 Nov |
1 |
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14698154 | Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with the antipsychotic drug sulpiride. | 2004 Jan 19 |
2 |
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15070333 | Designed, functionalized helix-loop-helix motifs that bind human carbonic anhydrase II: a new class of synthetic receptor molecules. | 2004 Apr 14 |
1 |
| 90 |
15081039 | Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with fluorine-containing sulfonamides. The first subnanomolar CA IX inhibitor discovered. | 2004 May 3 |
1 |
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15482952 | Carbonic anhydrase inhibitors: inhibition of human cytosolic isozyme II and mitochondrial isozyme V with a series of benzene sulfonamide derivatives. | 2004 Nov 15 |
1 |
| 92 |
15499997 | In vitro inhibition effects of some new sulfonamide inhibitors on human carbonic anhydrase I and II. | 2004 Jun |
2 |
| 93 |
16134002 | The cyclooxygenase-2 inhibitor celecoxib is a potent inhibitor of human carbonic anhydrase II. | 2004 Oct |
1 |
| 94 |
12873509 | Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with a bis-sulfonamide-two heads are better than one? | 2003 Aug 18 |
2 |
| 95 |
14611844 | Carbonic anhydrase inhibitors: inhibition of human and murine mitochondrial isozymes V with anions. | 2003 Sep 1 |
1 |
| 96 |
11310605 | Carbonic anhydrase inhibitors: sulfonamides as antitumor agents? | 2001 Mar |
1 |
| 97 |
11676494 | The catalytic properties of human carbonic anhydrase IX. | 2001 Nov 2 |
1 |
| 98 |
11807116 | Carbonic anhydrase activity in tissues of the icefish Chionodraco hamatus and of the red-blooded teleosts Trematomus bernacchii and Anguilla anguilla. | 2001 Nov |
1 |
| 99 |
10811034 | Carbonic anhydrase inhibitors; phosphoryl-sulfonamides--a new class of high affinity inhibitors of isozymes I and II. | 2000 |
1 |
| 100 |
10995069 | Carbonic anhydrase inhibitors: synthesis of sulfonamides incorporating 2,4,6-trisubstituted-pyridinium-ethylcarboxamido moieties possessing membrane-impermeability and in vivo selectivity for the membrane-bound (CA IV) versus the cytosolic (CA I and CA II) isozymes. | 2000 |
1 |