| 1 |
34596922 | Novel benzenesulfonamide-bearing pyrazoles and 1,2,4-thiadiazoles as selective carbonic anhydrase inhibitors. | 2022 Jan |
1 |
| 2 |
35489270 | Targeting the interplay between MMP-2, CA II and VEGFR-2 via new sulfonamide-tethered isomeric triazole hybrids; Microwave-assisted synthesis, computational studies and evaluation. | 2022 Jul |
2 |
| 3 |
35618035 | Nanozyme based on ZIF-8 for the colorimetric detection of sulfonamides in cow milk. | 2022 Sep 1 |
2 |
| 4 |
33038795 | Novel 3-substituted coumarins as selective human carbonic anhydrase IX and XII inhibitors: Synthesis, biological and molecular dynamics analysis. | 2021 Jan 1 |
1 |
| 5 |
34324968 | Novel carbohydrate-based sulfonamide derivatives as selective carbonic anhydrase II inhibitors: Synthesis, biological and molecular docking analysis. | 2021 Nov 1 |
1 |
| 6 |
34358123 | Synthesis and Human Carbonic Anhydrase I, II, IX, and XII Inhibition Studies of Sulphonamides Incorporating Mono-, Bi- and Tricyclic Imide Moieties. | 2021 Jul 19 |
1 |
| 7 |
34481530 | Inhibition of carbonic anhydrase II by sulfonamide derivatives. | 2021 Sep 1 |
2 |
| 8 |
34605430 | Determination of intracellular protein-ligand binding affinity by competition binding in-cell NMR. | 2021 Oct 1 |
1 |
| 9 |
34728369 | Discovery of novel aminosaccharide-based sulfonamide derivatives as potential carbonic anhydrase II inhibitors. | 2021 Dec 1 |
1 |
| 10 |
31718943 | Synthesis, biological and molecular dynamics investigations with a series of triazolopyrimidine/triazole-based benzenesulfonamides as novel carbonic anhydrase inhibitors. | 2020 Jan 1 |
1 |
| 11 |
31825195 | A New Strategy for Reporting Specific Protein Binding Events at Aqueous-Liquid Crystal Interfaces in the Presence of Non-Specific Proteins. | 2020 Feb 19 |
4 |
| 12 |
31911296 | Structure-activity relationship of human carbonic anhydrase-II inhibitors: Detailed insight for future development as anti-glaucoma agents. | 2020 Jan |
1 |
| 13 |
32182519 | Appliance of the piperidinyl-hydrazidoureido linker to benzenesulfonamide compounds: Synthesis, in vitro and in silico evaluation of potent carbonic anhydrase II, IX and XII inhibitors. | 2020 May |
1 |
| 14 |
32456080 | Synthetic Strategies and Computational Inhibition Activity Study for Triazinyl-Substituted Benzenesulfonamide Conjugates with Polar and Hydrophobic Amino Acids as Inhibitors of Carbonic Anhydrases. | 2020 May 22 |
1 |
| 15 |
32891000 | Pyridinium derivatives of 3-aminobenzenesulfonamide are nanomolar-potent inhibitors of tumor-expressed carbonic anhydrase isozymes CA IX and CA XII. | 2020 Oct |
1 |
| 16 |
30807935 | Synthesis of sulfonamide, amide and amine hybrid pharmacophore, an entry of new class of carbonic anhydrase II inhibitors and evaluation of chemo-informatics and binding analysis. | 2019 May |
2 |
| 17 |
30811749 | Investigation of the effects of some sulfonamides on acetylcholinesterase and carbonic anhydrase enzymes. | 2019 May |
1 |
| 18 |
31129502 | Synthesis, biological evaluation and in silico studies of novel N-substituted phthalazine sulfonamide compounds as potent carbonic anhydrase and acetylcholinesterase inhibitors. | 2019 Aug |
1 |
| 19 |
31136893 | Benzensulfonamides bearing spyrohydantoin moieties act as potent inhibitors of human carbonic anhydrases II and VII and show neuropathic pain attenuating effects. | 2019 Sep 1 |
1 |
| 20 |
31207328 | Chemometrical-electrochemical investigation for comparing inhibitory effects of quercetin and its sulfonamide derivative on human carbonic anhydrase II: Theoretical and experimental evidence. | 2019 Sep 1 |
3 |
| 21 |
31515058 | Synthesis and exploration of 2-morpholino-4-phenylthiazol-5-yl acrylamide derivatives for their effects against carbonic anhydrase I, II, IX and XII isoforms as a non-sulfonamide class of inhibitors. | 2019 Nov 1 |
1 |
| 22 |
29462772 | Design and synthesis of novel 1,3-diaryltriazene-substituted sulfonamides as potent and selective carbonic anhydrase II inhibitors. | 2018 Apr |
1 |
| 23 |
30176324 | Mechanistic investigation of sulfonamide ligands as human carbonic anhydrase II inhibitors. | 2018 Dec |
2 |
| 24 |
30253337 | Synthesis of different thio-scaffolds bearing sulfonamide with subnanomolar carbonic anhydrase II and IX inhibitory properties and X-ray investigations for their inhibitory mechanism. | 2018 Dec |
1 |
| 25 |
28110167 | Chiral separation of new sulfonamide derivatives and evaluation of their enantioselective affinity for human carbonic anhydrase II by microscale thermophoresis and surface plasmon resonance. | 2017 Apr 15 |
3 |
| 26 |
28111158 | Synthesis of isoxazole-containing sulfonamides with potent carbonic anhydrase II and VII inhibitory properties. | 2017 Feb 15 |
1 |
| 27 |
28753093 | Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo[d]thiazole-5- and 6-sulfonamides. | 2017 Dec |
1 |
| 28 |
26700575 | Kinetic and Structural Insights into the Mechanism of Binding of Sulfonamides to Human Carbonic Anhydrase by Computational and Experimental Studies. | 2016 May 12 |
2 |
| 29 |
26796953 | Sulfonamides incorporating heteropolycyclic scaffolds show potent inhibitory action against carbonic anhydrase isoforms I, II, IX and XII. | 2016 Feb 15 |
1 |
| 30 |
26810836 | Kinetic and X-ray crystallographic investigations on carbonic anhydrase isoforms I, II, IX and XII of a thioureido analog of SLC-0111. | 2016 Mar 1 |
3 |
| 31 |
27160030 | Isoform-selective inhibitory profile of 2-imidazoline-substituted benzene sulfonamides against a panel of human carbonic anhydrases. | 2016 |
1 |
| 32 |
27211329 | Carbonic anhydrase inhibition and the management of neuropathic pain. | 2016 Aug |
1 |
| 33 |
27234893 | Synthesis of 4-(thiazol-2-ylamino)-benzenesulfonamides with carbonic anhydrase I, II and IX inhibitory activity and cytotoxic effects against breast cancer cell lines. | 2016 Jul 1 |
2 |
| 34 |
27325502 | Label-enhanced surface plasmon resonance applied to label-free interaction analysis of small molecules and fragments. | 2016 Oct 1 |
1 |
| 35 |
27396930 | Synthesis 4-[2-(2-mercapto-4-oxo-4H-quinazolin-3-yl)-ethyl]-benzenesulfonamides with subnanomolar carbonic anhydrase II and XII inhibitory properties. | 2016 Sep 15 |
1 |
| 36 |
27435177 | Synthesis and carbonic anhydrase inhibitory activities of new thienyl-substituted pyrazoline benzenesulfonamides. | 2016 |
1 |
| 37 |
27474804 | Synthesis of novel bisindolylmethanes: New carbonic anhydrase II inhibitors, docking, and 3D pharmacophore studies. | 2016 Oct |
1 |
| 38 |
28002963 | Structure-Activity Relationship for Sulfonamide Inhibition of Helicobacter pylori α-Carbonic Anhydrase. | 2016 Dec 22 |
1 |
| 39 |
24666294 | Inhibition of human carbonic anhydrase isozymes I, II, IX and XII with a new series of sulfonamides incorporating aroylhydrazone-, [1,2,4]triazolo[3,4-b][1,3,4]thiadiazinyl- or 2-(cyanophenylmethylene)-1,3,4-thiadiazol-3(2H)-yl moieties. | 2015 Feb |
1 |
| 40 |
25733161 | X-ray crystallographic and kinetic investigations of 6-sulfamoyl-saccharin as a carbonic anhydrase inhibitor. | 2015 Apr 7 |
1 |
| 41 |
26160114 | Probing the 'bipolar' nature of the carbonic anhydrase active site: aromatic sulfonamides containing 1,3-oxazol-5-yl moiety as picomolar inhibitors of cytosolic CA I and CA II isoforms. | 2015 Aug 28 |
1 |
| 42 |
26199669 | Azobenzene-based inhibitors of human carbonic anhydrase II. | 2015 |
3 |
| 43 |
26534780 | Carbonic anhydrase inhibitors: Design, synthesis, kinetic, docking and molecular dynamics analysis of novel glycine and phenylalanine sulfonamide derivatives. | 2015 Dec 1 |
1 |
| 44 |
26639945 | Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activity. | 2015 Dec 15 |
1 |
| 45 |
23311862 | Carbonic anhydrase inhibitory properties of novel sulfonamide derivatives of aminoindanes and aminotetralins. | 2014 Feb |
1 |
| 46 |
24112770 | Discovering isozyme-selective inhibitor scaffolds of human carbonic anhydrases using structural alignment and de novo drug design approaches. | 2014 Feb |
1 |
| 47 |
24146387 | Glaucoma and the applications of carbonic anhydrase inhibitors. | 2014 |
1 |
| 48 |
25310626 | Structural insights on carbonic anhydrase inhibitory action, isoform selectivity, and potency of sulfonamides and coumarins incorporating arylsulfonylureido groups. | 2014 Nov 13 |
1 |
| 49 |
25358036 | A class of 4-sulfamoylphenyl-ω-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects. | 2014 Nov 26 |
1 |
| 50 |
25898725 | Comparison of QSAR models based on combinations of genetic algorithm, stepwise multiple linear regression, and artificial neural network methods to predict Kd of some derivatives of aromatic sulfonamides as carbonic anhydrase II inhibitors. | 2014 Jan-Feb |
1 |