Rimonabant

cannabinoid receptor 1 ; Homo sapiens







257 Article(s)
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201 15613777 New perspectives in the studies on endocannabinoid and cannabis: cannabinoid receptors and schizophrenia. 2004 Dec 1
202 20641388 (-)-3-(4-Chlorophenyl)-N'-[(4-[11C]cyanophenyl)sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine 2004 2
203 12399252 Anti-obesity effect of SR141716, a CB1 receptor antagonist, in diet-induced obese mice. 2003 Feb 1
204 12570386 Synthesis, structure-activity relationship, and evaluation of SR141716 analogues: development of central cannabinoid receptor ligands with lower lipophilicity. 2003 Feb 13 1
205 12690115 Hypersensitization of the Orexin 1 receptor by the CB1 receptor: evidence for cross-talk blocked by the specific CB1 antagonist, SR141716. 2003 Jun 27 5
206 12737320 Dual effect of cannabinoid CB1 receptor stimulation on a vanilloid VR1 receptor-mediated response. 2003 Mar 2
207 12759440 Subversion and utilization of the host cell cyclic adenosine 5'-monophosphate/protein kinase A pathway by Brucella during macrophage infection. 2003 Jun 1 2
208 12813001 Reduction of human monocytic cell neurotoxicity and cytokine secretion by ligands of the cannabinoid-type CB2 receptor. 2003 Jun 1
209 12823468 Anandamide regulates neuropeptide release from capsaicin-sensitive primary sensory neurons by activating both the cannabinoid 1 receptor and the vanilloid receptor 1 in vitro. 2003 Jun 1
210 12890515 Modulation of electrically evoked acetylcholine release through cannabinoid CB1 receptors: evidence for an endocannabinoid tone in the human neocortex. 2003 2
211 14561865 Biphasic effects of cannabinoids on acetylcholine release in the hippocampus: site and mechanism of action. 2003 Oct 15 1
212 14613317 An aromatic microdomain at the cannabinoid CB(1) receptor constitutes an agonist/inverse agonist binding region. 2003 Nov 20 2
213 14746372 Anandamide enhances extracellular levels of adenosine and induces sleep: an in vivo microdialysis study. 2003 Dec 15 1
214 12038810 Functional assessment of neuronal cannabinoid receptors in the muscular layers of human ileum and colon. 2002 Apr 1
215 12381672 Direct inhibition by cannabinoids of human 5-HT3A receptors: probable involvement of an allosteric modulatory site. 2002 Nov 1
216 12435794 N-(piperidin-1-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide (SR141716A) interaction with LYS 3.28(192) is crucial for its inverse agonism at the cannabinoid CB1 receptor. 2002 Dec 4
217 11236843 Effects of SR141716A on ethanol and sucrose self-administration. 2001 Feb 1
218 11296091 Blockade of effects of smoked marijuana by the CB1-selective cannabinoid receptor antagonist SR141716. 2001 Apr 3
219 11358910 Cannabinoids and the gastrointestinal tract. 2001 Jun 2
220 11397872 Normal human pituitary gland and pituitary adenomas express cannabinoid receptor type 1 and synthesize endogenous cannabinoids: first evidence for a direct role of cannabinoids on hormone modulation at the human pituitary level. 2001 Jun 1
221 11698062 The cannabinoid CB1 receptor antagonist SR 141716A reverses the antiemetic and motor depressant actions of WIN 55, 212-2. 2001 Oct 26 1
222 10614630 Suppression of nerve growth factor Trk receptors and prolactin receptors by endocannabinoids leads to inhibition of human breast and prostate cancer cell proliferation. 2000 Jan 1
223 10698714 Functional CB1 cannabinoid receptors in human vascular endothelial cells. 2000 Mar 15 1
224 10716447 Cannabinoids control spasticity and tremor in a multiple sclerosis model. 2000 Mar 2 1
225 10871313 CB1 cannabinoid receptor-mediated cell migration. 2000 Jul 1
226 10974429 Lack of response suppression follows repeated ventral tegmental cannabinoid administration: an in vitro electrophysiological study. 2000 1
227 11067978 Cannabinoid and kappa opioid receptors reduce potassium K current via activation of G(s) proteins in cultured hippocampal neurons. 2000 Nov 1
228 11081515 Bidirectional control of airway responsiveness by endogenous cannabinoids. 2000 Nov 2 1
229 9933150 Characterization of cannabinoid receptors coupled to vasorelaxation by endothelium-derived hyperpolarizing factor. 1999 Jan 2
230 10217281 Involvement of the carboxyl terminus of the third intracellular loop of the cannabinoid CB1 receptor in constitutive activation of Gs. 1999 May 2
231 10323591 Anandamide-induced mobilization of cytosolic Ca2+ in endothelial cells. 1999 Apr 1
232 10341254 Presynaptically located CB1 cannabinoid receptors regulate GABA release from axon terminals of specific hippocampal interneurons. 1999 Jun 1 1
233 10362691 Cannabinoid CB1 receptor of cat cerebral arterial muscle functions to inhibit L-type Ca2+ channel current. 1999 Jun 1
234 10392859 Finding of the endocannabinoid signalling system in Hydra, a very primitive organism: possible role in the feeding response. 1999 1
235 10394995 Blockade of cannabinoid (CB1) receptors by 141716 selectively antagonizes drug-induced reinstatement of exploratory behaviour in gerbils. 1999 May 1
236 10433501 Cannabinoid receptor activation inhibits GABAergic neurotransmission in rostral ventromedial medulla neurons in vitro. 1999 Jun 1
237 10469889 The development of cannabinoid antagonists. 1999 Aug 2
238 10493099 Cannabinoid modulation of dynorphin A: correlation to cannabinoid-induced antinociception. 1999 Aug 13 2
239 10494885 Presynaptic cannabinoid and imidazoline receptors in the human heart and their potential relationship. 1999 Aug 1
240 10531431 The CB1 cannabinoid receptor can sequester G-proteins, making them unavailable to couple to other receptors. 1999 Nov 1 1
241 10612710 Synergistic interactions of endogenous opioids and cannabinoid systems. 1999 Nov 27 1
242 11741201 Design and synthesis of the CB1 selective cannabinoid antagonist AM281: a potential human SPECT ligand. 1999 1
243 9653194 The endogenous cannabinoid anandamide inhibits human breast cancer cell proliferation. 1998 Jul 7 1
244 9685157 Control of pain initiation by endogenous cannabinoids. 1998 Jul 16 1
245 9688276 Biosynthesis and degradation of bioactive fatty acid amides in human breast cancer and rat pheochromocytoma cells--implications for cell proliferation and differentiation. 1998 Jun 15 1
246 9690851 Evidence for inverse agonism of SR141716A at human recombinant cannabinoid CB1 and CB2 receptors. 1998 Jun 4
247 9884065 In vitro functional evidence of neuronal cannabinoid CB1 receptors in human ileum. 1998 Dec 2
248 9126878 Receptor mediation in cannabinoid stimulated arachidonic acid mobilization and anandamide synthesis. 1997 1
249 9204917 Concurrent stimulation of cannabinoid CB1 and dopamine D2 receptors augments cAMP accumulation in striatal neurons: evidence for a Gs linkage to the CB1 receptor. 1997 Jul 15 2
250 9268384 A selective inverse agonist for central cannabinoid receptor inhibits mitogen-activated protein kinase activation stimulated by insulin or insulin-like growth factor 1. Evidence for a new model of receptor/ligand interactions. 1997 Aug 29 3