Rimonabant

cannabinoid receptor 1 ; Homo sapiens







257 Article(s)
Download
PMID
Title
Pub. Year
#Total Relationships
1 33573565 The Endocannabinoid System and Alcohol Dependence: Will Cannabinoid Receptor 2 Agonism be More Fruitful than Cannabinoid Receptor 1 Antagonism? 2022 2
2 32885412 Acute rimonabant treatment promotes protein synthesis in C2C12 myotubes through a CB1-independent mechanism. 2021 Apr 1
3 33931678 CB1 antagonism increases excitatory synaptogenesis in a cortical spheroid model of fetal brain development. 2021 Apr 30 1
4 34064024 Role of the Endocannabinoid System in the Adipose Tissue with Focus on Energy Metabolism. 2021 May 21 2
5 34326318 A novel chemical inhibitor suppresses breast cancer cell growth and metastasis through inhibiting HPIP oncoprotein. 2021 Jul 29 1
6 31917333 Δ9-tetrahydrocannabinol and 2-AG decreases neurite outgrowth and differentially affects ERK1/2 and Akt signaling in hiPSC-derived cortical neurons. 2020 Mar 1
7 31925452 The cannabinoid ligands SR141716A and AM251 enhance human and mouse islet function via GPR55-independent signalling. 2020 Nov 2
8 31981244 Rimonabant suppresses RNA transcription of hepatitis B virus by inhibiting hepatocyte nuclear factor 4α. 2020 May 1
9 32417279 Behavioral assessment of rimonabant under acute and chronic conditions. 2020 Jul 15 1
10 32512776 Targeting the Endocannabinoid CB1 Receptor to Treat Body Weight Disorders: A Preclinical and Clinical Review of the Therapeutic Potential of Past and Present CB1 Drugs. 2020 Jun 4 1
11 32927872 A Peripheral CB1R Antagonist Increases Lipolysis, Oxygen Consumption Rate, and Markers of Beiging in 3T3-L1 Adipocytes Similar to RIM, Suggesting that Central Effects Can Be Avoided. 2020 Sep 10 1
12 33002729 Chlorotrimethylsilane promoted one-flask heterocyclic synthesis of 1,2,4-triazoles from nitrilimines: Modeling studies and bioactivity evaluation of LH-21 and Rimonabant analogues. 2020 Nov 1
13 30649023 Cannabis effects on lipoproteins. 2019 Apr 1
14 30687889 Targeting CB1 and GPR55 Endocannabinoid Receptors as a Potential Neuroprotective Approach for Parkinson's Disease. 2019 Aug 2
15 31284863 Overcoming the Psychiatric Side Effects of the Cannabinoid CB1 Receptor Antagonists: Current Approaches for Therapeutics Development. 2019 1
16 31469511 The cannabinoid receptor 1 is involved in renal fibrosis during chronic allograft dysfunction: Proof of concept. 2019 Nov 1
17 31564385 Divalent cannabinoid-1 receptor ligands: A linker attachment point survey of SR141716A for development of high-affinity CB1R molecular probes. 2019 Nov 1 5
18 28661046 Activation of CaMKKβ/AMPKα pathway by 2-AG in human platelets. 2018 Jan 2
19 29407764 Rimonabant, a potent CB1 cannabinoid receptor antagonist, is a Gαi/o protein inhibitor. 2018 May 1 3
20 29417597 Acute Ethanol Inhibition of Adult Hippocampal Neurogenesis Involves CB1 Cannabinoid Receptor Signaling. 2018 Apr 2
21 29551963 Cannabinoid Receptors Modulate Excitation of an Olfactory Bulb Local Circuit by Cortical Feedback. 2018 2
22 29792186 Involvement of the CB2 cannabinoid receptor in cell growth inhibition and G0/G1 cell cycle arrest via the cannabinoid agonist WIN 55,212-2 in renal cell carcinoma. 2018 May 23 1
23 30077609 Synthesis and pharmacological characterization of functionalized 6-piperazin-1-yl-purines as cannabinoid receptor 1 (CB1) inverse agonists. 2018 Aug 15 1
24 30262909 Genetic and pharmacological regulation of the endocannabinoid CB1 receptor in Duchenne muscular dystrophy. 2018 Sep 27 1
25 30460698 Anandamide Induces Platelet Nitric Oxide Synthase through AMP-Activated Protein Kinase. 2018 Sep 1
26 28222356 Extinction of avoidance behavior by safety learning depends on endocannabinoid signaling in the hippocampus. 2017 Jul 1
27 28564576 The endocannabinoid system as a target for addiction treatment: Trials and tribulations. 2017 Sep 15 2
28 28947487 Cannabinoid CB1 Discrimination: Effects of Endocannabinoids and Catabolic Enzyme Inhibitors. 2017 Dec 1
29 29308855 [Prospects for the Use of Cannabinoid Receptor Ligands for the Treatment of Metabolic Syndrome and Atherosclerosis: Analysis of Experimental and Clinical Data]. 2017 1
30 29354056 Rimonabant Kills Colon Cancer Stem Cells without Inducing Toxicity in Normal Colon Organoids. 2017 1
31 26123153 Roles for the endocannabinoid system in ethanol-motivated behavior. 2016 Feb 4 2
32 26803499 Self-administration of the anandamide transport inhibitor AM404 by squirrel monkeys. 2016 May 1
33 27208730 Hierarchical glucocorticoid-endocannabinoid interplay regulates the activation of the nucleus accumbens by insulin. 2016 Jun 1
34 25411367 (4-(Bis(4-fluorophenyl)methyl)piperazin-1-yl)(cyclohexyl)methanone hydrochloride (LDK1229): a new cannabinoid CB1 receptor inverse agonist from the class of benzhydryl piperazine analogs. 2015 Feb 4
35 25859226 Role of the endogenous cannabinoid system in nicotine addiction: novel insights. 2015 2
36 25893829 Anti Proliferative and Pro Apoptotic Effects of Flavonoid Quercetin Are Mediated by CB1 Receptor in Human Colon Cancer Cell Lines. 2015 Dec 1
37 26008966 Cannabinoid receptor CB1 regulates STAT3 activity and its expression dictates the responsiveness to SR141716 treatment in human glioma patients' cells. 2015 Jun 20 4
38 26157624 Influence of rimonabant treatment on peripheral blood mononuclear cells; flow cytometry analysis and gene expression profiling. 2015 2
39 26362774 The CB1 Neutral Antagonist Tetrahydrocannabivarin Reduces Default Mode Network and Increases Executive Control Network Resting State Functional Connectivity in Healthy Volunteers. 2015 Sep 10 1
40 26365347 N-Oleoyl glycine, a lipoamino acid, stimulates adipogenesis associated with activation of CB1 receptor and Akt signaling pathway in 3T3-L1 adipocyte. 2015 Oct 23 1
41 23452341 The hepatic cannabinoid 1 receptor as a modulator of hepatic energy state and food intake. 2014 Jan 1
42 24366865 Allosteric modulation of a cannabinoid G protein-coupled receptor: binding site elucidation and relationship to G protein signaling. 2014 Feb 28 1
43 24467410 Cannabinoids inhibit cholinergic contraction in human airways through prejunctional CB1 receptors. 2014 Jun 1
44 24692267 Involvement of cannabinoid receptor-1 activation in mitochondrial depolarizing effect of lipopolysaccharide in human spermatozoa. 2014 Jul 1
45 24747288 Prospective therapeutic agents for obesity: molecular modification approaches of centrally and peripherally acting selective cannabinoid 1 receptor antagonists. 2014 May 22 1
46 25096297 Design, synthesis and in vitro evaluation of novel uni- and bivalent ligands for the cannabinoid receptor type 1 with variation of spacer length and structure. 2014 Sep 1 1
47 25713910 Rimonabant inhibits proliferation, collagen secretion and induces apoptosis in hepatic stellate cells. 2014 Oct 3
48 23070073 Neutral antagonism at the cannabinoid 1 receptor: a safer treatment for obesity. 2013 Dec 1
49 23278450 LiCABEDS II. Modeling of ligand selectivity for G-protein-coupled cannabinoid receptors. 2013 Jan 28 2
50 23287700 Cannabinoid discrimination and antagonism by CB(1) neutral and inverse agonist antagonists. 2013 Mar 1