Acetazolamide

carbonic anhydrase 1 ; Homo sapiens







30 Article(s)
Download
PMID
Title
Pub. Year
#Total Relationships
1 34385868 Novel Mannich bases with strong carbonic anhydrases and acetylcholinesterase inhibition effects: 3-(aminomethyl)-6-{3-[4-(trifluoromethyl)phenyl]acryloyl}-2(3H)-benzoxazolones. 2021 2
2 34387019 Inhibition Profiles of Some Symmetric Sulfamides Derived from Phenethylamines on Human Carbonic Anhydrase I, and II Isoenzymes. 2021 Oct 1
3 31887473 Synthesis and selective inhibitory effects of some 2-oxindole benzenesulfonamide conjugates on human carbonic anhydrase isoforms CA I, CA II, CA IX and CAXII. 2020 Jan 1
4 30597695 Evaluation of antimicrobial, antibiofilm and carbonic anhydrase inhibition profiles of 1,3-bis-chalcone derivatives. 2019 Apr 1
5 28792233 Synthesis of chalcone-imide derivatives and investigation of their anticancer and antimicrobial activities, carbonic anhydrase and acetylcholinesterase enzymes inhibition profiles. 2018 Feb 1
6 29149534 Novel N-propylphthalimide- and 4-vinylbenzyl-substituted benzimidazole salts: Synthesis, characterization, and determination of their metal chelating effects and inhibition profiles against acetylcholinesterase and carbonic anhydrase enzymes. 2018 Jan 1
7 29283199 Synthesis and investigation of the conversion reactions of pyrimidine-thiones with nucleophilic reagent and evaluation of their acetylcholinesterase, carbonic anhydrase inhibition, and antioxidant activities. 2018 Feb 1
8 27780313 Synthesis, carbonic anhydrase I and II isoenzymes inhibition properties, and antibacterial activities of novel tetralone-based 1,4-benzothiazepine derivatives. 2017 Apr 1
9 27984137 Novel eugenol derivatives: Potent acetylcholinesterase and carbonic anhydrase inhibitors. 2017 Jan 1
10 28065499 Benzenesulfonamide bearing imidazothiadiazole and thiazolotriazole scaffolds as potent tumor associated human carbonic anhydrase IX and XII inhibitors. 2017 Feb 1 2
11 28100082 Synthesis and bioactivity of several new hetaryl sulfonamides. 2017 Dec 1
12 28117934 Synthesis of new cyclic thioureas and evaluation of their metal-chelating activity, acetylcholinesterase, butyrylcholinesterase, and carbonic anhydrase inhibition profiles. 2017 Jul 2
13 28544359 Discovery of potent carbonic anhydrase, acetylcholinesterase, and butyrylcholinesterase enzymes inhibitors: The new amides and thiazolidine-4-ones synthesized on an acetophenone base. 2017 Sep 1
14 27050248 Synthesis of some tetrahydropyrimidine-5-carboxylates, determination of their metal chelating effects and inhibition profiles against acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase. 2016 Dec 1
15 27075164 The synthesis of some β-lactams and investigation of their metal-chelating activity, carbonic anhydrase and acetylcholinesterase inhibition profiles. 2016 1
16 27579806 Synthesis, cytotoxicity and carbonic anhydrase inhibitory activities of new pyrazolines. 2016 2
17 24758348 Intrinsic thermodynamics of sulfonamide inhibitor binding to human carbonic anhydrases I and II. 2015 Apr 1
18 26105196 Sulfonamide bearing pyrazolylpyrazolines as potent inhibitors of carbonic anhydrase isoforms I, II, IX and XII. 2015 Aug 15 1
19 26459317 CA1 contributes to microcalcification and tumourigenesis in breast cancer. 2015 Oct 12 1
20 25456084 4-Functionalized 1,3-diarylpyrazoles bearing 6-aminosulfonylbenzothiazole moiety as potent inhibitors of carbonic anhydrase isoforms hCA I, II, IX and XII. 2014 Dec 15 2
21 22733110 Polypharmacology of sulfonamides: pazopanib, a multitargeted receptor tyrosine kinase inhibitor in clinical use, potently inhibits several mammalian carbonic anhydrases. 2012 Aug 25 1
22 22838845 Carbonic anhydrase I (CA1) is involved in the process of bone formation and is susceptible to ankylosing spondylitis. 2012 Jul 27 1
23 20553118 Synthesis of 5-amino-1,3,4-thiadiazole-2-sulphonamide derivatives and their inhibition effects on human carbonic anhydrase isozymes. 2011 Apr 1
24 18336307 The alpha and beta classes carbonic anhydrases from Helicobacter pylori as novel drug targets. 2008 1
25 15110853 Carbonic anhydrase inhibitors: aromatic and heterocyclic sulfonamides incorporating adamantyl moieties with strong anticonvulsant activity. 2004 May 15 1
26 11430635 Indomethacin activates carbonic anhydrase and antagonizes the effect of the specific carbonic anhydrase inhibitor acetazolamide, by a direct mechanism of action. 2001 Jun 1
27 10768298 Topiramate as an inhibitor of carbonic anhydrase isoenzymes. 2000 2
28 11140609 Carbonic anhydrase inhibitors: synthesis of Schiff bases of hydroxybenzaldehydes with aromatic sulfonamides and their reactions with arylsulfonyl isocyanates. 2000 1
29 8667211 Nonsteroidal anti-inflammatory drugs activate carbonic anhydrase by a direct mechanism of action. 1996 Jun 2
30 6430170 Inactive form of carbonic anhydrase I in erythrocytes from primary aldosteronism. 1984 2