PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 30902024-12 2020 CYP2C19 inhibitor (+)-N-3-benzylnirvanol and CYP3A inhibitor ketoconazole significantly reduced microsomal normeperidine generation by an individual donor with high CYP2C19 activity, whereas donors with lower CYP2C19 activity were sensitive to inhibition by ketoconazole but not benzylnirvanol. Ketoconazole 61-73 cytochrome P450 family 3 subfamily A member 4 Homo sapiens 45-50 30902024-12 2020 CYP2C19 inhibitor (+)-N-3-benzylnirvanol and CYP3A inhibitor ketoconazole significantly reduced microsomal normeperidine generation by an individual donor with high CYP2C19 activity, whereas donors with lower CYP2C19 activity were sensitive to inhibition by ketoconazole but not benzylnirvanol. Ketoconazole 258-270 cytochrome P450 family 3 subfamily A member 4 Homo sapiens 45-50