PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 34676043-0 2021 Amino-Heterocycle Tetrahydroisoquinoline CXCR4 Antagonists with Improved ADME Profiles via Late-Stage Buchwald Couplings. 1,2,3,4-tetrahydroisoquinoline 18-40 chemokine (C-X-C motif) receptor 4 Mus musculus 41-46 30052039-0 2018 Design, Synthesis, and Pharmacological Evaluation of Second-Generation Tetrahydroisoquinoline-Based CXCR4 Antagonists with Favorable ADME Properties. 1,2,3,4-tetrahydroisoquinoline 71-93 chemokine (C-X-C motif) receptor 4 Mus musculus 100-105 30052039-3 2018 We previously disclosed a hit-to-lead effort that led to the discovery of a series of tetrahydroisoquinoline-based CXCR4 antagonists exemplified by the lead compound TIQ15. 1,2,3,4-tetrahydroisoquinoline 86-108 chemokine (C-X-C motif) receptor 4 Mus musculus 115-120