PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 23689570-10 2013 NF-kappaB is regulated by the proteasome and saquinavir, a HIV protease inhibitor, is provided with antiproteasome activity. Saquinavir 45-55 nuclear factor kappa B subunit 1 Homo sapiens 0-9 22431705-5 2012 The effects of saquinavir on NF-kappaB nuclear localization in cultured PBMCs and in immortalized human podocytes were assessed. Saquinavir 15-25 nuclear factor kappa B subunit 1 Homo sapiens 29-38 22431705-10 2012 In culture, saquinavir blunted NF-kappaB activation in human podocytes and in PBMCs. Saquinavir 12-22 nuclear factor kappa B subunit 1 Homo sapiens 31-40 12234989-5 2002 For this reason, we investigated whether the HIV-I protease inhibitor saquinavir can inhibit NF-kappaB activation, block 26s proteasome activity in prostate cancer cells, and promote their apoptosis. Saquinavir 70-80 nuclear factor kappa B subunit 1 Homo sapiens 93-102 12234989-6 2002 The effect of saquinavir on LPS/IFN-gamma-induced activation of NF-kappaB was assessed by gel-shift assays and by Western analysis of corresponding IkappaBalpha-levels. Saquinavir 14-24 nuclear factor kappa B subunit 1 Homo sapiens 64-73 12234989-9 2002 Saquinavir treatment prevented LPS/IFN-gamma-induced activation of NF-kappaB in RAW cells and stabilized expression of IkappaBalpha. Saquinavir 0-10 nuclear factor kappa B subunit 1 Homo sapiens 67-76