PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 33332480-3 2020 Upadacitinib tartrate (Rinvoq), a selective and reversible JAK1 inhibitor, inhibited interleukin (IL)-6 and IL-7 and ameliorated adjuvant-induced arthritis in preclinical studies. upadacitinib 23-29 interleukin 6 Homo sapiens 85-103 31448433-2 2020 This study characterizes the relationships between upadacitinib exposure and interleukin (IL)-6-induced signal transducer and activator of transcription proteins 3 (STAT3) phosphorylation (pSTAT3) and IL-7-induced STAT5 phosphorylation (pSTAT5) in the ex vivo setting as measures for JAK1 and JAK1/JAK3 inhibition, respectively, with comparison to tofacitinib. upadacitinib 51-63 interleukin 6 Homo sapiens 77-95 31448433-5 2020 Upadacitinib (and tofacitinib) reversibly inhibited IL-6-induced pSTAT3 and IL-7-induced pSTAT5 in a concentration-dependent manner. upadacitinib 0-12 interleukin 6 Homo sapiens 52-56