PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 25914645-7 2015 SLC22A1 IC50 values for efavirenz, darunavir, and prazosin were determined. efavirenz 24-33 solute carrier family 22 member 1 Homo sapiens 0-7 25914645-8 2015 Cellular accumulation of efavirenz and darunavir was also assessed in SLC22A1-expressing KCL22 cells and reversibility of this accumulation was assessed using prazosin. efavirenz 25-34 solute carrier family 22 member 1 Homo sapiens 70-77 25914645-11 2015 Absolute SLC22A1 IC50 values for efavirenz, darunavir, and prazosin were 21.8, 46.2, and 2.8 muM, respectively. efavirenz 33-42 solute carrier family 22 member 1 Homo sapiens 9-16 25914645-12 2015 Efavirenz accumulation was higher in SLC22A1-expressing cells compared to mock-transfected cells (17% higher, p = 0.009) which was reversed using prazosin, whereas no difference was observed for darunavir (p = 0.86). efavirenz 0-9 solute carrier family 22 member 1 Homo sapiens 37-44