PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 20870034-1 2010 KMUP-1 inhibits monocrotaline (MCT)-induced pulmonary artery (PA) proliferation by targeting serotonin (5-HT) receptors, inactivating RhoA and reducing phosphorylation of AKT/ERK. Monocrotaline 16-29 AKT serine/threonine kinase 1 Homo sapiens 171-174 20870034-1 2010 KMUP-1 inhibits monocrotaline (MCT)-induced pulmonary artery (PA) proliferation by targeting serotonin (5-HT) receptors, inactivating RhoA and reducing phosphorylation of AKT/ERK. Monocrotaline 31-34 AKT serine/threonine kinase 1 Homo sapiens 171-174 20870034-10 2010 In conclusion, KMUP-1 inhibits MCT-induced PA proliferation by binding to 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors, increasing endothelial eNOS/5-HT(2B) receptor expression and NO release and inhibiting 5-HTT/RhoA/ROCK expression and AKT/ERK phosphorylation. Monocrotaline 31-34 AKT serine/threonine kinase 1 Homo sapiens 235-238