PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 31514980-3 2019 The lowest IC50 was 12.9 micromol L-1 of anisodine on OCT1 and the highest was 1.8 mmol L-1 of monocrotaline on OCT2. Monocrotaline 95-108 solute carrier family 22 member 2 Homo sapiens 112-116 31514980-5 2019 Monocrotaline was determined to be a substrate of both OCT1 (Km = 109.1 +- 17.8 micromol L-1, Vmax = 576.5 +- 87.5 pmol/mg protein/min) and OCT2 (Km = 64.7 +- 14.8 micromol L-1, Vmax = 180.7 +- 22.0 pmol/mg protein/min), other than OCT3 and MATE transporters. Monocrotaline 0-13 solute carrier family 22 member 2 Homo sapiens 140-144