PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 27581642-0 2016 Structure-Activity Relationship Study of N(6)-Benzoyladenine-Type BRD4 Inhibitors and Their Effects on Cell Differentiation and TNF-alpha Production. N6-benzoyladenine 41-60 bromodomain containing 4 Homo sapiens 66-70 27581642-4 2016 We have reported potent N(6)-benzoyladenine-based inhibitors of BRD4, a BET family member that serves as a key mediator of transcriptional elongation. N6-benzoyladenine 24-43 bromodomain containing 4 Homo sapiens 64-68 25678016-0 2015 Discovery and structure-activity relationship studies of N6-benzoyladenine derivatives as novel BRD4 inhibitors. N6-benzoyladenine 57-74 bromodomain containing 4 Homo sapiens 96-100 25678016-3 2015 As a part of our continuing structural development studies of thalidomide to obtain a broad spectrum of biological modifiers based on the "multi-template" approach, in this work we focused on BRD4-inhibitory activity, and discovered that N6-benzoyladenine derivatives exhibit this activity. N6-benzoyladenine 238-255 bromodomain containing 4 Homo sapiens 192-196 25678016-5 2015 N6-Benzoyladenine appears to be a new chemical scaffold for development of BRD4 inhibitors. N6-benzoyladenine 0-17 bromodomain containing 4 Homo sapiens 75-79