PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 33262250-9 2021 Clofarabine and cladribine were ENT1 and ENT2 substrates, while nevirapine and lexibulin were ENT1 and ENT2 non-transported inhibitors. Cladribine 16-26 solute carrier family 29 member 1 (Augustine blood group) Homo sapiens 32-36 34894346-4 2022 Intestinal absorption and distribution of cladribine throughout the body appear to be essentially mediated by equilibrative NTs (ENTs) and concentrative NTs (CNTs), specifically by ENT1, ENT2, ENT4, CNT2 (low affinity), and CNT3. Cladribine 42-52 solute carrier family 29 member 1 (Augustine blood group) Homo sapiens 181-185 34894346-6 2022 A key transporter for the intracellular uptake of cladribine into B and T-lymphocytes is ENT1 with ancillary contributions of ENT2 and CNT2. Cladribine 50-60 solute carrier family 29 member 1 (Augustine blood group) Homo sapiens 89-93 34435310-6 2021 Intestinal absorption, distribution throughout the body, and intracellular uptake of cladribine appear to be exclusively mediated by equilibrative and concentrative nucleoside transporters, specifically by ENT1, ENT2, ENT4, CNT2 (low affinity), and CNT3. Cladribine 85-95 solute carrier family 29 member 1 (Augustine blood group) Homo sapiens 206-210 34435310-7 2021 Renal excretion of cladribine appears to be most likely driven by breast cancer resistance protein, ENT1, and P-glycoprotein. Cladribine 19-29 solute carrier family 29 member 1 (Augustine blood group) Homo sapiens 100-104 16234483-5 2006 When Cl-F-ara-A transport rates by hENT1 were compared with those of Cl-dAdo and F-ara-A, Cl-dAdo had the highest efficiency of transport, although Cl-F-ara-A showed the greatest accumulation during 5-min exposures. Cladribine 90-97 solute carrier family 29 member 1 (Augustine blood group) Homo sapiens 35-40 16234483-8 2006 Affinity studies with recombinant transporters produced in yeast showed that hENT1, hENT2, and hCNT3 all had higher affinities for Cl-F-ara-A than for either Cl-dAdo or F-ara-A. Cladribine 158-165 solute carrier family 29 member 1 (Augustine blood group) Homo sapiens 77-82 29987837-12 2019 Cladribine distribution across membranes is primarily facilitated by equilibrative nucleoside transporter (ENT) 1, concentrative nucleoside transporter (CNT) 3 and breast cancer resistance protein (BCRP), and there is no evidence of any cladribine-related effect on heart rate, atrioventricular conduction or cardiac repolarisation (QTc interval prolongation). Cladribine 0-10 solute carrier family 29 member 1 (Augustine blood group) Homo sapiens 69-113 16333246-7 2005 hENT1 mRNA expression also seemed to correlate inversely with the LC50 values of cladribine (rp=-0.30; P=0.04), decitabine (rp=-0.29; P=0.04) and gemcitabine (rp=-0.33; P=0.02). Cladribine 81-91 solute carrier family 29 member 1 (Augustine blood group) Homo sapiens 0-5