Title : Species differences in stereoselective metabolism of mephenytoin by cytochrome P450 (CYP2C and CYP3A).

Pub. Date : 1993 Jan

PMID : 8423554






2 Functional Relationships(s)
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1 Antibodies raised against CYP3A2 (anti-CYP3A) clearly inhibited microsomal 4"-hydroxylation of R-mephenytoin, but marginally S-mephenytoin, in rats. (R)-(-)-Mephenytoin cytochrome P450, family 3, subfamily a, polypeptide 2 Rattus norvegicus
2 Antibodies raised against CYP3A2 (anti-CYP3A) clearly inhibited microsomal 4"-hydroxylation of R-mephenytoin, but marginally S-mephenytoin, in rats. Mephenytoin cytochrome P450, family 3, subfamily a, polypeptide 2 Rattus norvegicus