Title : Chimeric constructs between human and rat equilibrative nucleoside transporters (hENT1 and rENT1) reveal hENT1 structural domains interacting with coronary vasoactive drugs.

Pub. Date : 1998 Aug 21

PMID : 9705281






1 Functional Relationships(s)
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Protein Name
Organism
1 hENT1 is also potently inhibited by coronary vasodilator drugs (dipyridamole, dilazep, and draflazine), whereas rENT1 is insensitive to inhibition by these compounds (dipyridamole IC50 values 190 nM (hENT1) and >/=10 microM (rENT1) at 10 microM uridine). draflazine solute carrier family 29 member 1 (Augustine blood group) Homo sapiens