Title : Esmolol, an ultrashort-acting, selective beta 1-adrenoceptor antagonist: pharmacodynamic and pharmacokinetic properties.

Pub. Date : 1994

PMID : 7957532






2 Functional Relationships(s)
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1 Up to a rate of infusion of esmolol of 500 micrograms.kg-1 BW.min-1 there was a maximal beta 1-receptor occupancy of 84.7% while beta 2-receptor occupancy was below the detection limit; confirming the beta 1 selectivity of esmolol. esmolol potassium calcium-activated channel subfamily M regulatory beta subunit 1 Homo sapiens
2 Up to a rate of infusion of esmolol of 500 micrograms.kg-1 BW.min-1 there was a maximal beta 1-receptor occupancy of 84.7% while beta 2-receptor occupancy was below the detection limit; confirming the beta 1 selectivity of esmolol. esmolol potassium calcium-activated channel subfamily M regulatory beta subunit 1 Homo sapiens