Pub. Date : 1995 Feb 14
PMID : 7768260
1 Functional Relationships(s)Download |
Sentence | Compound Name | Protein Name | Organism |
1 | [3H]BQ-123 binding was sensitive to endothelin-1 and endothelin-2 (Ki values = 0.058 and 0.10 nM, respectively) and the endothelin ETA receptor-selective antagonist BQ-123 (Ki = 3.3 nM), while showing low affinity for endothelin-3 (Ki = 50 nM), the endothelin ETB receptor-selective agonist BQ-3020 (Ki = 970 nM) and other bioactive peptides. | Tritium | endothelin 1 | Homo sapiens |