Title : Rifampicin induction of lidocaine metabolism in cultured human hepatocytes.

Pub. Date : 1995 Aug

PMID : 7636727






1 Functional Relationships(s)
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1 Rifampicin has been shown to induce CYP3A4, a major human hepatic CYP isozyme that is known to metabolize lidocaine to its primary metabolite, monoethylglycinexylidide. Lidocaine cytochrome P450 family 3 subfamily A member 4 Homo sapiens