Title : Sex and Estrous Cycle Differences in Analgesia and Brain Oxycodone Levels.

Pub. Date : 2021 Dec

PMID : 34581987






2 Functional Relationships(s)
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1 Propranolol (a CYP2D mechanism-based inhibitor), versus vehicle pre-treatments, increased brain oxycodone, and decreased brain oxymorphone/oxycodone drug level ratios (an in vivo CYP2D activity phenotype in the brain) in males and females in estrus, but not in females in diestrus. Propranolol cytochrome P450 family 2 subfamily D member 6 Homo sapiens
2 Propranolol (a CYP2D mechanism-based inhibitor), versus vehicle pre-treatments, increased brain oxycodone, and decreased brain oxymorphone/oxycodone drug level ratios (an in vivo CYP2D activity phenotype in the brain) in males and females in estrus, but not in females in diestrus. Propranolol cytochrome P450 family 2 subfamily D member 6 Homo sapiens