Title : Inhibition of CYP3A7 DHEA-S Oxidation by Lopinavir and Ritonavir: An Alternative Mechanism for Adrenal Impairment in HIV Antiretroviral-Treated Neonates.

Pub. Date : 2021 Apr 19

PMID : 33821626






1 Functional Relationships(s)
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1 Furthermore, ritonavir is a time-dependent inhibitor of CYP3A7 with a KI of 0.392 muM and a kinact of 0.119 min-1, illustrating the potential for CYP3A mediated drug-drug interactions with Kaletra. Ritonavir cytochrome P450 family 3 subfamily A member 4 Homo sapiens