Title : An acetyl-histone vulnerability in PI3K/AKT inhibition-resistant cancers is targetable by both BET and HDAC inhibitors.

Pub. Date : 2021 Feb 16

PMID : 33596421






2 Functional Relationships(s)
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1 Here, we demonstrate that PI3K/AKT inhibitors cause glycolytic crisis, acetyl-coenzyme A (CoA) shortage, and a global decrease in histone acetylation. Acetyl Coenzyme A AKT serine/threonine kinase 1 Homo sapiens
2 Here, we demonstrate that PI3K/AKT inhibitors cause glycolytic crisis, acetyl-coenzyme A (CoA) shortage, and a global decrease in histone acetylation. Acetyl Coenzyme A AKT serine/threonine kinase 1 Homo sapiens