Title : Characterization of interactions between local anesthetics and histamine H1 receptor by cell membrane chromatography model.

Pub. Date : 2021 Mar 20

PMID : 33497977






2 Functional Relationships(s)
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1 Results showed that the local anesthetics can directly occupy histamine binding sites on H1R, and the KD values obtained from different CMC methods exhibited positive correlations with each other (p < 0.01). Histamine histamine receptor H1 Homo sapiens
2 This was not only in line with the Ca2+ responses in activating H1R, but also consistent with the same amino acid residues shared with histamine in the H1R active site. Histamine histamine receptor H1 Homo sapiens