Pub. Date : 2021 Jan 8
PMID : 33420359
2 Functional Relationships(s)Download |
Sentence | Compound Name | Protein Name | Organism |
| 1 | A capsaicinoid-based soft drug, AG1529, for attenuating TRPV1-mediated histaminergic and inflammatory sensory neuron excitability. | Capsaicin | transient receptor potential cation channel subfamily V member 1 | Homo sapiens |
| 2 | We report that AG1529 competitively blocked capsaicin-evoked activation of hTRPV1 with micromolar potency, moderately affected pH-induced gating, and did not alter voltage- and heat-mediated responses. | Capsaicin | transient receptor potential cation channel subfamily V member 1 | Homo sapiens |