Title : High-dose etoposide formulations do not saturate intestinal P-glycoprotein: Development, stability, and pharmacokinetics in Sprague-Dawley rats.

Pub. Date : 2020 Jun 15

PMID : 32376439






1 Functional Relationships(s)
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1 The present study investigated if the BCS IV drug substance etoposide could be solubilized to a concentration saturating P-gp after oral administration. Etoposide ATP-binding cassette, subfamily B (MDR/TAP), member 1B Rattus norvegicus