Title : Evaluation of the Role of P-glycoprotein (P-gp)-Mediated Efflux in the Intestinal Absorption of Common Substrates with Elacridar, a P-gp Inhibitor, in Rats.

Pub. Date : 2020 Jun

PMID : 32078103






2 Functional Relationships(s)
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1 BACKGROUND AND OBJECTIVES: P-glycoprotein (P-gp) has been shown previously to contribute to the intestinal absorption of verapamil, diltiazem, tacrolimus, colchicine and indinavir in situ; however, its contribution in vivo is unknown. Diltiazem ATP-binding cassette, subfamily B (MDR/TAP), member 1B Rattus norvegicus
2 BACKGROUND AND OBJECTIVES: P-glycoprotein (P-gp) has been shown previously to contribute to the intestinal absorption of verapamil, diltiazem, tacrolimus, colchicine and indinavir in situ; however, its contribution in vivo is unknown. Diltiazem ATP-binding cassette, subfamily B (MDR/TAP), member 1B Rattus norvegicus