Title : p27 allosterically activates cyclin-dependent kinase 4 and antagonizes palbociclib inhibition.

Pub. Date : 2019 Dec 13

PMID : 31831640






1 Functional Relationships(s)
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1 We found that p27, when phosphorylated by tyrosine kinases, allosterically activated CDK4 in complex with cyclin D1 (CDK4-CycD1). Tyrosine cyclin D1 Homo sapiens