Title : Leprosy drug clofazimine activates peroxisome proliferator-activated receptor-γ and synergizes with imatinib to inhibit chronic myeloid leukemia cells.

Pub. Date : 2020 Apr

PMID : 31371410






2 Functional Relationships(s)
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1 Peroxisome proliferator-activated receptor-gamma (PPARgamma) agonist pioglitazone downregulates signal transducer and activator of transcription 5 (STAT5) and in combination with imatinib induces complete molecular response in imatinib-refractory patients by eroding leukemia stem cells. Imatinib Mesylate signal transducer and activator of transcription 5A Homo sapiens
2 Peroxisome proliferator-activated receptor-gamma (PPARgamma) agonist pioglitazone downregulates signal transducer and activator of transcription 5 (STAT5) and in combination with imatinib induces complete molecular response in imatinib-refractory patients by eroding leukemia stem cells. Imatinib Mesylate signal transducer and activator of transcription 5A Homo sapiens