Title : Leprosy drug clofazimine activates peroxisome proliferator-activated receptor-γ and synergizes with imatinib to inhibit chronic myeloid leukemia cells.

Pub. Date : 2020 Apr

PMID : 31371410






1 Functional Relationships(s)
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1 Combining imatinib with clofazimine caused a far superior synergy than pioglitazone where clofazimine reduced imatinib"s IC50 by >4 logs and remarkably eroded quiescent CD34+ cells. Imatinib Mesylate CD34 molecule Homo sapiens