Title : Inhibition of the mTOR pathway: A new mechanism of β cell toxicity induced by tacrolimus.

Pub. Date : 2019 Dec

PMID : 31152486






5 Functional Relationships(s)
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Compound Name
Protein Name
Organism
1 Tacrolimus (TAC) and rapamycin (Rapa) both bind to FK506-binding protein 12 (FKBP12). Tacrolimus FKBP prolyl isomerase 1A Rattus norvegicus
2 Tacrolimus (TAC) and rapamycin (Rapa) both bind to FK506-binding protein 12 (FKBP12). Tacrolimus FKBP prolyl isomerase 1A Rattus norvegicus
3 Tacrolimus (TAC) and rapamycin (Rapa) both bind to FK506-binding protein 12 (FKBP12). Tacrolimus FKBP prolyl isomerase 1A Rattus norvegicus
4 Tacrolimus (TAC) and rapamycin (Rapa) both bind to FK506-binding protein 12 (FKBP12). Tacrolimus FKBP prolyl isomerase 1A Rattus norvegicus
5 In silico docking and immunoprecipitation experiments confirmed that TAC can form a stable noncovalent interaction with FKBP12-mTOR. Tacrolimus FKBP prolyl isomerase 1A Rattus norvegicus