Title : Discovery of Quinazolin-4(3 H)-ones as NLRP3 Inflammasome Inhibitors: Computational Design, Metal-Free Synthesis, and in Vitro Biological Evaluation.

Pub. Date : 2019 May 3

PMID : 30896160






1 Functional Relationships(s)
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1 The nitro-substituted quinazolin-4(3 H)-one 2k inhibited NLRP3 inflammasome (IC50 5 muM) via the suppression of IL-1beta release from ATP-stimulated J774A.1 cells. Adenosine Triphosphate interleukin 1 beta Mus musculus