Title : Csk-homologous kinase (Chk) is an efficient inhibitor of Src-family kinases but a poor catalyst of phosphorylation of their C-terminal regulatory tyrosine.

Pub. Date : 2017 Aug 7

PMID : 28784162






1 Functional Relationships(s)
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1 RESULTS: Our results revealed Csk as a robust enzyme catalysing phosphorylation of the C-terminal tail tyrosine of SFKs but a weak non-catalytic inhibitor of SFKs. Tyrosine C-terminal Src kinase Homo sapiens