Title : Functionalized PLA-PEG nanoparticles targeting intestinal transporter PepT1 for oral delivery of acyclovir.

Pub. Date : 2017 Aug 30

PMID : 28705621






2 Functional Relationships(s)
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1 In Caco-2 cell monolayer model, competition between functionalized nanoparticles and [3H]Glycylsarcosine, a strong substrate of PepT1, reduced [3H]Glycylsarcosine transport from 22 to 46%. Tritium solute carrier family 15 member 1 Homo sapiens
2 In Caco-2 cell monolayer model, competition between functionalized nanoparticles and [3H]Glycylsarcosine, a strong substrate of PepT1, reduced [3H]Glycylsarcosine transport from 22 to 46%. Tritium solute carrier family 15 member 1 Homo sapiens