Title : Association of NR1I2, CYP3A5 and ABCB1 genetic polymorphisms with variability of temsirolimus pharmacokinetics and toxicity in patients with metastatic bladder cancer.

Pub. Date : 2017 Sep

PMID : 28676933






2 Functional Relationships(s)
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1 The metabolism of temsirolimus and its active metabolite sirolimus mainly depends on cytochrome P450 3A4/5 (CYP3A4/A5) and the ABCB1 transporter. Sirolimus cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 The metabolism of temsirolimus and its active metabolite sirolimus mainly depends on cytochrome P450 3A4/5 (CYP3A4/A5) and the ABCB1 transporter. Sirolimus cytochrome P450 family 3 subfamily A member 4 Homo sapiens