Pub. Date : 2017 Dec
PMID : 28417439
2 Functional Relationships(s)Download |
Sentence | Compound Name | Protein Name | Organism |
1 | Clinical Pharmacokinetics of Sacubitril/Valsartan (LCZ696): A Novel Angiotensin Receptor-Neprilysin Inhibitor. | Valsartan | membrane metalloendopeptidase | Homo sapiens |
2 | Absorption of sacubitril/valsartan and conversion of sacubitril (prodrug) to sacubitrilat (neprilysin inhibitor) was rapid with maximum plasma concentrations of sacubitril, sacubitrilat, and valsartan (angiotensin receptor blocker) reaching within 0.5, 1.5-2.0, and 2.0-3.0 h, respectively. | Valsartan | membrane metalloendopeptidase | Homo sapiens |