Title : Semisimultaneous Midazolam Administration to Evaluate the Time Course of CYP3A Activation by a Single Oral Dose of Efavirenz.

Pub. Date : 2017 Jul

PMID : 28194792






1 Functional Relationships(s)
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1 In 12 healthy participants individual CYP3A activity was quantified using a semisimultaneous methodology (midazolam orally and 6 hours later intravenously) both alone and during a period of 22 days after a single oral dose of 400 mg efavirenz. efavirenz cytochrome P450 family 3 subfamily A member 4 Homo sapiens