Title : Planarian cholinesterase: in vitro characterization of an evolutionarily ancient enzyme to study organophosphorus pesticide toxicity and reactivation.

Pub. Date : 2017 Aug

PMID : 27990564






1 Functional Relationships(s)
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Protein Name
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1 Inhibition by classic protonable amine and quaternary reversible inhibitors (ethopropazine, donepezil, tacrine, edrophonium, BW284c51, propidium) shows that DjChE is far less sensitive to these inhibitors than human AChE, suggesting discrete differences in active center and peripheral site recognition and structures. Propidium acetylcholinesterase (Cartwright blood group) Homo sapiens