Title : BRET-based β-arrestin2 recruitment to the histamine H1 receptor for investigating antihistamine binding kinetics.

Pub. Date : 2016 Sep

PMID : 27468652






1 Functional Relationships(s)
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1 Antihistamines displayed similar kinetic signatures on antagonizing histamine-induced beta-arrestin2 recruitment as compared to displacing radioligand binding from the H1R. Histamine histamine receptor H1 Homo sapiens