Title : Nitroimidazole carboxamides as antiparasitic agents targeting Giardia lamblia, Entamoeba histolytica and Trichomonas vaginalis.

Pub. Date : 2016 Sep 14

PMID : 27236016






2 Functional Relationships(s)
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1 Several of the new compounds exhibited potent activity against G. lamblia strains, including metronidazole-resistant strains of G. lamblia (EC50 = 0.1-2.5 muM cf. Metronidazole latexin Homo sapiens
2 metronidazole EC50 = 6.1-18 muM). Metronidazole latexin Homo sapiens